SCHEMBL22014739

SCHEMBL22014739

CC(C)c1cc2c(c(C(C)C)c1CC(N)=O)OC(F)(F)O2

nearest known ligand 0.33

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
NLRP3 Q96P20 1/20 0.33
SIRT1 Q96EB6 2/20 0.32
GABRA1 P14867 1/20 0.30
GABRG2 P18507 1/20 0.30
GABRB3 P28472 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30276820 1.00 NLRP3 (0.33) NLRP3SIRT1GABRA1GABRG2GABRB3
SCHEMBL21962160 0.88 KDM4E (0.33) NLRP3GABRA1GABRG2GABRB3
SCHEMBL21962238 0.87 NLRP3 (0.33) NLRP3GABRA1GABRG2GABRB3
SCHEMBL22014365 0.86 NLRP3 (0.38) NLRP3GABRA1GABRG2GABRB3
SCHEMBL20698765 0.72 SIRT1 (0.35) NLRP3SIRT1
SCHEMBL16843335 0.70
SCHEMBL20028908 0.70 GABRA1 (0.30) GABRA1GABRG2GABRB3
SCHEMBL20698736 0.69 NLRP3 (0.40) NLRP3SIRT1
SCHEMBL8859174 0.68 FABP3 (0.33)
SCHEMBL24192685 0.67 ADORA2A (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020102574-A1 THE COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH NLRP ACTIVITY NOVARTIS INFLAMMASOME RESEARCH, INC. (US) 2020-05-22 WO disclosed