SCHEMBL22014446

SCHEMBL22014446

CCc1cc(C#N)cc(C(C)C)c1CC(=O)/N=C(\N)c1ccc(CN(C)C)cc1

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NLRP3 Q96P20 1/20 0.33
HRH3 Q9Y5N1 1/20 0.33
NSD2 O96028 1/20 0.33
ROCK2 O75116 1/20 0.33
CYP2D6 P10635 1/20 0.32
CYP2C19 P33261 1/20 0.32
OPRK1 P41145 1/20 0.32
HSP90AA1 P07900 2/20 0.31
LSS P48449 1/20 0.31
GSR P00390 1/20 0.30
SLC6A2 P23975 1/20 0.30
SLC6A4 P31645 1/20 0.30
SLC6A3 Q01959 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25139315 0.85 NLRP3 (0.33) NLRP3ROCK2CYP2D6CYP2C19LSS
SCHEMBL20698683 0.83 NLRP3 (0.39) NLRP3ROCK2CYP2D6CYP2C19OPRK1
SCHEMBL22014445 0.83 NLRP3 (0.39) NLRP3ROCK2CYP2D6CYP2C19OPRK1
SCHEMBL22014582 0.82 NLRP3 (0.34) NLRP3ROCK2LSSGSR
SCHEMBL20698684 0.81 NLRP3 (0.33) NLRP3ROCK2LSSGSR
SCHEMBL25067186 0.81 NLRP3 (0.39) NLRP3OPRK1LSS
SCHEMBL23692211 0.79 ROCK2 (0.35) NLRP3ROCK2CYP2D6LSS
SCHEMBL20698800 0.78 NLRP3 (0.38) NLRP3ROCK2LSS
SCHEMBL22014583 0.77 NLRP3 (0.42) NLRP3NSD2ROCK2OPRK1HSP90AA1
SCHEMBL20698687 0.77 NLRP3 (0.42) NLRP3NSD2ROCK2OPRK1HSP90AA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020102574-A1 THE COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH NLRP ACTIVITY NOVARTIS INFLAMMASOME RESEARCH, INC. (US) 2020-05-22 WO disclosed