SCHEMBL22014502

SCHEMBL22014502

CCN(CCN(CCNC[C@H](C)O)C[C@H](C)O)Cc1ccc(C(=O)NCP(=O)(O)O)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRK1 P41145 7/20 0.42
OPRM1 P35372 5/20 0.42
HDAC8 Q9BY41 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
LMNA P02545 2/20 0.39
ALDH1A1 P00352 2/20 0.39
SLC22A2 O15244 1/20 0.39
SLC22A1 O15245 1/20 0.39
TSHR P16473 1/20 0.39
ACHE P22303 1/20 0.39
MAPK1 P28482 1/20 0.39
CYP2C19 P33261 1/20 0.39
BLM P54132 2/20 0.38
PMP22 Q01453 1/20 0.38
SCN1A P35498 1/20 0.38
SCN2A Q99250 1/20 0.38
SCN3A Q9NY46 1/20 0.38
NFKB1 P19838 1/20 0.37
KCNH2 Q12809 1/20 0.37
POLB P06746 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22014321 0.90 OPRK1 (0.39) OPRK1OPRM1HDAC8HDAC6LMNA
SCHEMBL22014325 0.87 OPRK1 (0.42) OPRK1OPRM1HDAC8HDAC6LMNA
SCHEMBL24672619 0.84 HDAC8 (0.41) OPRK1OPRM1HDAC8HDAC6ALDH1A1
SCHEMBL22014463 0.83 OPRK1 (0.44) OPRK1OPRM1ALDH1A1MAPK1SMN1; SMN2
SCHEMBL22014497 0.81 PTPN1 (0.44) OPRK1OPRM1HDAC8HDAC6CA12
SCHEMBL22014501 0.79 PTPN1 (0.60) OPRK1OPRM1LMNACA12CA9
SCHEMBL24672243 0.78 PYCR1 (0.33) HDAC8HDAC6ALDH1A1TSHRPOLB
SCHEMBL22014453 0.77 OPRK1 (0.38) OPRK1OPRM1TSHRATMSMN1; SMN2
SCHEMBL24672914 0.77 POLB (0.44) OPRK1OPRM1TSHRMAPK1POLB
SCHEMBL22014469 0.76 CA2 (0.44) OPRK1OPRM1CA12CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020102820-A1 COMPOUNDS FOR USE AS IRON (III) MRI CONTRAST AGENTS CONTAINING ANIONIC PENDENTS AND ANCILLARY GROUPS THE RESEARCH FOUNDATION FOR THE STATE UNIVERSITY OF NEW YORK (US) 2020-05-22 WO disclosed