SCHEMBL22014810

SCHEMBL22014810

C[C@@]12CNC[C@]1(C)CN(c1ccc(N3CCSCC3)cc1)C2

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.49
MAPT P10636 3/20 0.49
LGMN Q99538 2/20 0.46
ADRB1 P08588 6/20 0.39
AKR1C3 P42330 1/20 0.37
HTR3E A5X5Y0 4/20 0.36
HTR3B O95264 4/20 0.36
HTR3A P46098 4/20 0.36
HTR3D Q70Z44 4/20 0.36
HTR3C Q8WXA8 4/20 0.36
SIGMAR1 Q99720 4/20 0.36
THRB P10828 1/20 0.36
SIRT6 Q8N6T7 1/20 0.34
APP P05067 1/20 0.33
TSHR P16473 2/20 0.33
USP2 O75604 2/20 0.33
CYP2D6 P10635 2/20 0.33
TP53 P04637 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22015789 0.80 ALDH1A1 (0.50) ALDH1A1MAPTLGMNADRB1THRB
SCHEMBL27400025 0.77 ADRB1 (0.53) ALDH1A1MAPTADRB1AKR1C3SIGMAR1
SCHEMBL22014811 0.76 KDM4E (0.50) ALDH1A1ADRB1HTR3EHTR3BHTR3A
SCHEMBL25387770 0.76 ALDH1A1 (0.42) ALDH1A1MAPTTSHRUSP2TP53
SCHEMBL22015091 0.75 ADRB1 (0.36) ALDH1A1MAPTADRB1HTR3EHTR3B
SCHEMBL22015092 0.73 HIF1A (0.50) ALDH1A1MAPTTHRBTSHRUSP2
SCHEMBL8648308 0.72 ADRB1 (0.57) ALDH1A1MAPTLGMNADRB1AKR1C3
SCHEMBL21963849 0.71 ALDH1A1 (0.57) ALDH1A1MAPTTSHRUSP2CYP2D6
SCHEMBL12490848 0.70 ALDH1A1 (0.56) ALDH1A1MAPTLGMNAKR1C3THRB
SCHEMBL20907841 0.69 ADRB1 (0.53) ALDH1A1MAPTADRB1HTR3EHTR3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020099886-A1 LOX INHIBITORS THE INSTITUTE OF CANCER RESEARCH: ROYAL CANCER HOSPITAL (GB) 2020-05-22 WO disclosed