SCHEMBL22015091

SCHEMBL22015091

C[S+]([O-])N1CCN(c2ccc(N3C[C@]4(C)CNC[C@]4(C)C3)cc2)CC1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB1 P08588 5/20 0.36
HTR3A P46098 4/20 0.36
HTR3E A5X5Y0 3/20 0.36
HTR3B O95264 3/20 0.36
HTR3D Q70Z44 3/20 0.36
HTR3C Q8WXA8 3/20 0.36
SIGMAR1 Q99720 3/20 0.36
HTR5A P47898 1/20 0.36
SIRT6 Q8N6T7 2/20 0.35
KDM4E B2RXH2 3/20 0.33
KMT2A Q03164 3/20 0.33
ALDH1A1 P00352 2/20 0.33
GAA P10253 2/20 0.33
MAPT P10636 2/20 0.33
PTK2B Q14289 2/20 0.33
ADRA2C P18825 1/20 0.33
GFER P55789 1/20 0.33
ESR2 Q92731 1/20 0.33
MEN1 O00255 2/20 0.32
LMNA P02545 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17642641 0.78 MEN1 (0.50) ADRB1KMT2AALDH1A1MAPTMEN1
SCHEMBL22015789 0.76 ALDH1A1 (0.50) ADRB1KDM4EKMT2AALDH1A1GAA
SCHEMBL22537561 0.76 AKR1C3 (0.42) ADRB1HTR3ASIRT6KDM4EKMT2A
SCHEMBL22014810 0.75 ALDH1A1 (0.49) ADRB1HTR3AHTR3EHTR3BHTR3D
SCHEMBL17320506 0.73 KDM4E (0.46) KDM4EKMT2AALDH1A1GAAMAPT
SCHEMBL22015092 0.73 HIF1A (0.50) KDM4EKMT2AALDH1A1GAAMAPT
SCHEMBL22014811 0.72 KDM4E (0.50) ADRB1HTR3AHTR3EHTR3BHTR3D
SCHEMBL25387770 0.72 ALDH1A1 (0.42) KDM4EKMT2AALDH1A1GAAMAPT
SCHEMBL19491900 0.68 SIRT6 (0.44) SIRT6KDM4EKMT2AALDH1A1GAA
SCHEMBL4519141 0.66 ADRB1 (0.58) ADRB1HTR3AHTR3EHTR3BHTR3D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020099886-A1 LOX INHIBITORS THE INSTITUTE OF CANCER RESEARCH: ROYAL CANCER HOSPITAL (GB) 2020-05-22 WO disclosed