SCHEMBL22015250

SCHEMBL22015250

CC(=O)N[C@@H]1C(=O)N2C(C(=O)O)=C(COC(=O)c3cn(C4CC4)c4cc(N5CCNCC5)c(F)cc4c3=O)CSC12

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.55
ALDH1A1 P00352 4/20 0.55
LMNA P02545 3/20 0.55
HPGD P15428 3/20 0.55
HSD17B10 Q99714 3/20 0.55
CYP1A2 P05177 1/20 0.55
TOP2A P11388 1/20 0.55
CYP2C9 P11712 1/20 0.55
TOP2B Q02880 1/20 0.55
MAPT P10636 2/20 0.48
PIK3CG P48736 3/20 0.43
PIK3CD O00329 1/20 0.43
PIK3R1 P27986 1/20 0.43
PIK3CA P42336 1/20 0.43
BRD4 O60885 1/20 0.42
TSHR P16473 1/20 0.42
HTT P42858 1/20 0.42
CYP2J2 P51589 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
L3MBTL1 Q9Y468 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22014780 1.00 KDM4E (0.55) KDM4EALDH1A1LMNAHPGDHSD17B10
SCHEMBL22014785 0.92 KDM4E (0.55) KDM4EALDH1A1LMNAHPGDHSD17B10
SCHEMBL8498659 0.91 KDM4E (0.55) KDM4EALDH1A1LMNAHPGDHSD17B10
SCHEMBL21963921 0.89 ALDH1A1 (0.49) KDM4EALDH1A1LMNAHPGDHSD17B10
SCHEMBL22015249 0.89 HPGD (0.54) KDM4EALDH1A1LMNAHPGDHSD17B10
SCHEMBL22014786 0.89 ALDH1A1 (0.49) KDM4EALDH1A1LMNAHPGDHSD17B10
SCHEMBL22015248 0.89 HPGD (0.54) KDM4EALDH1A1LMNAHPGDHSD17B10
SCHEMBL21964156 0.89 TOP2B (0.49) KDM4EALDH1A1LMNAHPGDHSD17B10
SCHEMBL10379270 0.88 KDM4E (0.49) KDM4EALDH1A1LMNAHPGDHSD17B10
SCHEMBL22015246 0.86 HPGD (0.47) KDM4EALDH1A1LMNAHPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020099858-A1 CEPHALOSPORIN CIPROFLOXACIN HYBRID COMPOUNDS IMPERIAL COLLEGE OF SCIENCE, TECHNOLOGY AND MEDICINE (GB) 2020-05-22 WO disclosed