SCHEMBL2201861

SCHEMBL2201861

O=C(OOC(=O)C1CCC1)C1CCC1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.54
HTT P42858 1/20 0.54
KMT2A Q03164 1/20 0.54
TDP1 Q9NUW8 1/20 0.54
CES2 O00748 1/20 0.45
CES1 P23141 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.41
CHRM2 P08172 2/20 0.39
CHRM4 P08173 2/20 0.39
CHRM1 P11229 2/20 0.39
CHRM3 P20309 2/20 0.39
MIF P14174 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
NOS2 P35228 1/20 0.36
ALDH1A1 P00352 2/20 0.36
TSHR P16473 1/20 0.36
RECQL P46063 1/20 0.36
POLB P06746 1/20 0.35
ATM Q13315 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2202711 0.93 CES2 (0.53) SMN1; SMN2HTTKMT2ATDP1CES2
SCHEMBL2198986 0.90 CES2 (0.58) SMN1; SMN2HTTKMT2ATDP1CES2
SCHEMBL29281908 0.87
SCHEMBL2197391 0.86 KMT2A (0.40) SMN1; SMN2HTTKMT2ATDP1CES2
SCHEMBL6113076 0.84 SMN1; SMN2 (0.52) SMN1; SMN2HTTKMT2ATDP1CES2
SCHEMBL573198 0.83 CES2 (0.50) SMN1; SMN2HTTKMT2ATDP1CES2
SCHEMBL28209666 0.81
SCHEMBL30068399 0.81 ALDH1A1 (0.42) SMN1; SMN2HTTKMT2ATDP1ALDH1A1
SCHEMBL382048 0.81 SMN1; SMN2 (0.41) SMN1; SMN2HTTKMT2ATDP1CES2
SCHEMBL1481528 0.79

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 20 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7740826-B2 Method for functionalizing carbon nanotubes utilizing peroxides WILLIAM MARSH RICE UNIVERSITY (US) 2010-06-22 US claimed
US-20090306427-A1 Chemical Functionalization of Carbon Nanotubes NATIONAL RESEARCH COUNCIL OF CANADA (CA) 2009-12-10 US claimed
EP-1989143-A1 CHEMICAL FUNCTIONALIZATION OF CARBON NANOTUBES National Research Council of Canada (CA) 2008-11-12 EP claimed
WO-2007098578-A1 CHEMICAL FUNCTIONALIZATION OF CARBON NANOTUBES NATIONAL RESEARCH COUNCIL OF CANADA (CA) 2007-09-07 WO claimed
US-20070098620-A1 Method for functionalizing carbon nanotubes utilizing peroxides WILLIAM MARSH RICE UNIVERSITY (US) 2007-05-03 US claimed
US-20040223900-A1 Method for functionalizing carbon nanotubes utilizing peroxides WILLIAM MARSH RICE UNIVERSITY (US) 2004-11-11 US claimed
EP-3087060-B1 PYRIMIDONE CARBOXAMIDE COMPOUNDS AS PDE2 INHIBITORS MERCK SHARP & DOHME (US) 2020-05-13 EP disclosed
US-9815796-B2 Pyrimidone carboxamide compounds as PDE2 inhibitors MERCK SHARP & DOHME CORP. (US) 2017-11-14 US disclosed
US-20170015633-A1 PYRIMIDONE CARBOXAMIDE COMPOUNDS AS PDE2 INHIBITORS MERCK SHARP & DOHME CORP. (US) 2017-01-19 US disclosed
EP-3087060-A1 PYRIMIDONE CARBOXAMIDE COMPOUNDS AS PDE2 INHIBITORS Merck Sharp & Dohme Corp. (US) 2016-11-02 EP disclosed
WO-2015096651-A1 PYRIMIDONE CARBOXAMIDE COMPOUNDS AS PDE2 INHIBITORS MERCK SHARP & DOHME CORP. (US) 2015-07-02 WO disclosed
US-7976816-B2 Method for functionalizating carbon naontubes utilizing peroxides WILLIAM MARSH RICE UNIVERSITY (US) 2011-07-12 US disclosed
US-20100222536-A1 Method for Functionalizating Carbon Naontubes Utilizing Peroxides WILLIAM MARSH RICE UNIVERSITY (US) 2010-09-02 US disclosed
US-7740826-B2 Method for functionalizing carbon nanotubes utilizing peroxides WILLIAM MARSH RICE UNIVERSITY (US) 2010-06-22 US disclosed
US-20090306427-A1 Chemical Functionalization of Carbon Nanotubes NATIONAL RESEARCH COUNCIL OF CANADA (CA) 2009-12-10 US disclosed
EP-1989143-A1 CHEMICAL FUNCTIONALIZATION OF CARBON NANOTUBES National Research Council of Canada (CA) 2008-11-12 EP disclosed
WO-2007098578-A1 CHEMICAL FUNCTIONALIZATION OF CARBON NANOTUBES NATIONAL RESEARCH COUNCIL OF CANADA (CA) 2007-09-07 WO disclosed
US-20070098620-A1 Method for functionalizing carbon nanotubes utilizing peroxides WILLIAM MARSH RICE UNIVERSITY (US) 2007-05-03 US disclosed
US-7125533-B2 decomposing an acyl peroxide to form carbon-centered free radicals and reacting the carbon-centered free radicals with the carbon nanotube to form a functionalized carbon nanotube WILLIAM MARSH RICE UNIVERSITY (US) 2006-10-24 US disclosed
US-20040223900-A1 Method for functionalizing carbon nanotubes utilizing peroxides WILLIAM MARSH RICE UNIVERSITY (US) 2004-11-11 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170015633-A1 PYRIMIDONE CARBOXAMIDE COMPOUNDS AS PDE2 INHIBITORS PDE2A, PDE12, PDE3A SMN1; SMN2 204/4885HTT 4240/4885KMT2A 1732/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.