SCHEMBL22018853

SCHEMBL22018853

CCN1CCC(CC(=O)NCc2cc(Cl)cc(Cl)c2)CC1

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 3/20 0.50
NPC1 O15118 2/20 0.50
GHSR Q92847 1/20 0.46
EPHX1 P07099 1/20 0.45
CACNA1I Q9P0X4 7/20 0.45
KCNH2 Q12809 5/20 0.45
HRH3 Q9Y5N1 1/20 0.43
ERCC1 P07992 1/20 0.42
ERCC4 Q92889 1/20 0.42
ENPP2 Q13822 1/20 0.42
DRD2 P14416 1/20 0.41
DRD3 P35462 1/20 0.41
TP53 P04637 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
MAPK1 P28482 1/20 0.41
POLB P06746 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22019050 0.85 CACNA1I (0.48) RAB9ANPC1CACNA1IKCNH2ERCC1
SCHEMBL22019049 0.84 CACNA1I (0.47) RAB9ANPC1CACNA1IKCNH2ERCC1
SCHEMBL4273159 0.82 CACNA1I (0.49) RAB9ANPC1CACNA1IKCNH2ENPP2
SCHEMBL19112992 0.81 CACNA1I (0.47) RAB9ANPC1CACNA1IKCNH2ENPP2
SCHEMBL19112805 0.81 CACNA1I (0.48) RAB9ANPC1CACNA1IKCNH2ENPP2
SCHEMBL4270993 0.79 CACNA1I (0.45) RAB9ANPC1CACNA1IKCNH2CYP2D6
SCHEMBL22019051 0.79 NPC1 (0.42) RAB9ANPC1CACNA1IKCNH2ENPP2
SCHEMBL4278734 0.78 CACNA1I (0.43) RAB9ANPC1CACNA1IKCNH2ENPP2
SCHEMBL4275836 0.78 CACNA1I (0.46) RAB9ANPC1CACNA1IKCNH2ENPP2
SCHEMBL4269196 0.78 CACNA1I (0.46) RAB9ANPC1CACNA1IKCNH2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3189839-B1 N-PIPERIDINYL ACETAMIDE DERIVATIVES AS CALCIUM CHANNEL BLOCKERS PRAXIS PREC MEDICINES INC (US) 2020-05-20 EP disclosed