SCHEMBL22019151

SCHEMBL22019151

CS(=O)(=O)c1cccc(C(=O)c2cnc(N3CCCC3c3ccccn3)s2)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KRAS P01116 1/20 0.41
KDM4A O75164 1/20 0.41
KDM4B O94953 1/20 0.41
KDM5C P41229 1/20 0.41
KDM5B Q9UGL1 1/20 0.41
NUDT1 P36639 2/20 0.39
TSHR P16473 2/20 0.38
LMNA P02545 1/20 0.38
GCK P35557 1/20 0.37
HTT P42858 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
ROCK2 O75116 1/20 0.36
VNN1 O95497 4/20 0.35
MAP4K1 Q92918 1/20 0.35
PIK3C3 Q8NEB9 2/20 0.35
PRMT5 O14744 1/20 0.35
WDR77 Q9BQA1 1/20 0.35
MLYCD O95822 1/20 0.35
HDAC8 Q9BY41 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21962448 1.00 KRAS (0.41) KRASKDM4AKDM4BKDM5CKDM5B
SCHEMBL21962682 0.88 NR1H2 (0.39) ROCK2MLYCD
SCHEMBL22019320 0.88 NR1H2 (0.39) ROCK2MLYCD
SCHEMBL21962690 0.86 CPT2 (0.39) TSHRLMNAHTTMLYCD
SCHEMBL22019317 0.86 CPT2 (0.39) TSHRLMNAHTTMLYCD
SCHEMBL22019319 0.85 VNN1 (0.42) NUDT1TSHRLMNAVNN1
SCHEMBL21962626 0.85 VNN1 (0.42) NUDT1TSHRLMNAVNN1
SCHEMBL22020535 0.84 VNN1 (0.44) ROCK2VNN1MLYCDHDAC8HDAC6
SCHEMBL21962341 0.84 VNN1 (0.44) ROCK2VNN1MLYCDHDAC8HDAC6
SCHEMBL22020531 0.83 GRM5 (0.43) NUDT1GCKHTTVNN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020102575-A1 HETEROCYCLIC AMINOTHIAZOLES AND USES THEREOF INCEPTION IBD, INC. (US) 2020-05-22 WO disclosed