SCHEMBL22019319

SCHEMBL22019319

CS(=O)(=O)c1cccc(C(=O)c2cnc(N3CCCC3c3cccnc3)s2)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
VNN1 O95497 1/20 0.42
ALDH1A1 P00352 6/20 0.42
KDM4E B2RXH2 3/20 0.42
LMNA P02545 2/20 0.41
MAPT P10636 2/20 0.41
SCN9A Q15858 3/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C19 P33261 1/20 0.41
BLM P54132 1/20 0.40
ALOX15 P16050 1/20 0.40
CHRNA7 P36544 2/20 0.40
CHRNB2 P17787 2/20 0.40
CHRNB4 P30926 2/20 0.40
CHRNA3 P32297 2/20 0.40
CHRNA4 P43681 2/20 0.40
CHRNA2 Q15822 2/20 0.40
TDP1 Q9NUW8 2/20 0.40
HTR3E A5X5Y0 1/20 0.40
PSIP1 O75475 1/20 0.40
TRPA1 O75762 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21962626 1.00 VNN1 (0.42) VNN1ALDH1A1KDM4ELMNAMAPT
SCHEMBL21962682 0.91 NR1H2 (0.39) SCN9A
SCHEMBL22019320 0.91 NR1H2 (0.39) SCN9A
SCHEMBL21962690 0.89 CPT2 (0.39) LMNATSHR
SCHEMBL22019317 0.89 CPT2 (0.39) LMNATSHR
SCHEMBL22020535 0.87 VNN1 (0.44) VNN1SCN9ATRPA1
SCHEMBL21962341 0.87 VNN1 (0.44) VNN1SCN9ATRPA1
SCHEMBL22019151 0.85 KRAS (0.41) VNN1LMNATSHRNUDT1
SCHEMBL21962448 0.85 KRAS (0.41) VNN1LMNATSHRNUDT1
SCHEMBL22019146 0.83 VNN1 (0.42) VNN1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020102575-A1 HETEROCYCLIC AMINOTHIAZOLES AND USES THEREOF INCEPTION IBD, INC. (US) 2020-05-22 WO disclosed