SCHEMBL22020362

SCHEMBL22020362

Cc1nc2c(c(NC(N)=O)c1C1CC1)CCC2

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.43
CYP1A2 P05177 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
USP2 O75604 1/20 0.43
KDM4E B2RXH2 3/20 0.42
MAPT P10636 2/20 0.42
MEN1 O00255 1/20 0.40
TSHR P16473 1/20 0.40
KMT2A Q03164 1/20 0.40
EEF2K O00418 1/20 0.39
NLRP3 Q96P20 2/20 0.39
EHMT2 Q96KQ7 2/20 0.38
ACHE P22303 4/20 0.37
TDP1 Q9NUW8 1/20 0.36
HTT P42858 1/20 0.34
LMNA P02545 1/20 0.33
SPR P35270 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21963067 0.89 GAA (0.46) GAACYP1A2NPSR1USP2KDM4E
SCHEMBL25821017 0.85 NLRP3 (0.50) GAACYP1A2NPSR1USP2KDM4E
SCHEMBL25838016 0.81 GAA (0.43) GAACYP1A2NPSR1USP2KDM4E
SCHEMBL22019806 0.79 GAA (0.59) GAACYP1A2NPSR1USP2KDM4E
SCHEMBL22020723 0.78 CYP1A2 (0.39) GAACYP1A2NPSR1USP2KDM4E
SCHEMBL30162291 0.78 CYP1A2 (0.39) GAACYP1A2NPSR1USP2KDM4E
SCHEMBL21963248 0.76 EEF2K (0.39) GAACYP1A2NPSR1USP2KDM4E
SCHEMBL22021099 0.74 NLRP3 (0.48) GAACYP1A2NPSR1USP2KDM4E
SCHEMBL22021144 0.74 NLRP3 (0.48) GAACYP1A2NPSR1USP2KDM4E
SCHEMBL22020326 0.73 ACHE (0.50) KDM4EMEN1KMT2AEEF2KACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020102096-A1 COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH NLRP ACTIVITY NOVARTIS INFLAMMASOME RESEARCH, INC. (US) 2020-05-22 WO disclosed
US-20160248025-A1 Organic Electroluminescent Device UDC IRELAND LTD (IE) 2016-08-25 US disclosed