Biphenyl

Biphenyl

SCHEMBL2202263

NC(=O)n1cnnn1.c1ccc(-c2ccccc2)cc1

nearest known ligand 0.44

Full drug profile on Sugi Atlas →

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.44
ALDH1A1 P00352 2/20 0.41
NPSR1 Q6W5P4 1/20 0.41
KMT2A Q03164 3/20 0.41
RAB9A P51151 2/20 0.41
SMN1; SMN2 Q16637 3/20 0.40
BCAT2 O15382 1/20 0.39
HMOX1 P09601 1/20 0.39
SCN4A P35499 1/20 0.38
TP53 P04637 1/20 0.38
KCNJ1 P48048 1/20 0.38
KDM4E B2RXH2 1/20 0.38
MEN1 O00255 1/20 0.38
HPGD P15428 1/20 0.37
ACLY P53396 1/20 0.37
GAA P10253 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL707611 0.84
SCHEMBL918756 0.74 NOTUM (0.47) NOTUMALDH1A1NPSR1KMT2ARAB9A
SCHEMBL4592417 0.72 MCL1 (0.41) NOTUMKMT2ARAB9ASMN1; SMN2HMOX1
SCHEMBL4592415 0.72 MCL1 (0.41) NOTUMKMT2ARAB9ASMN1; SMN2HMOX1
SCHEMBL1502065 0.70 KMT2A (0.50) NOTUMALDH1A1KMT2ASMN1; SMN2TP53
SCHEMBL3079013 0.70 TP53 (0.54) ALDH1A1KMT2ARAB9ASMN1; SMN2TP53
SCHEMBL4502875 0.69
Biphenyl SCHEMBL473288 0.68 ALDH1A1 (0.60) ALDH1A1SMN1; SMN2BCAT2KDM4EGAA
Biphenyl SCHEMBL335359 0.68 ALDH1A1 (0.60) ALDH1A1SMN1; SMN2BCAT2KDM4EGAA
Biphenyl SCHEMBL4593266 0.68 ALDH1A1 (0.60) ALDH1A1SMN1; SMN2BCAT2KDM4EGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2205573-B1 TETRAZOLE-SUBSTITUTED ARYL AMIDE DERIVATIVES AND USES THEREOF HOFFMANN LA ROCHE (CH) 2013-10-23 EP disclosed
US-7981914-B2 Tetrazole-substituted aryl amide derivatives and uses thereof ROCHE PALO ALTO LLC (US) 2011-07-19 US disclosed
EP-2205573-A1 TETRAZOLE-SUBSTITUTED ARYL AMIDE DERIVATIVES AND USES THEREOF F. Hoffmann-Roche AG (CH) 2010-07-14 EP disclosed
US-20090093523-A1 Tetrazole-substituted aryl amide derivatives and uses thereof ROCHE PALO ALTO LLC 2009-04-09 US disclosed
WO-2009043780-A1 TETRAZOLE-SUBSTITUTED ARYL AMIDE DERIVATIVES AND USES THEREOF F. HOFFMANN-LA ROCHE AG (CH) 2009-04-09 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090093523-A1 Tetrazole-substituted aryl amide derivatives and uses thereof AR, NAT1, TBXA2R NOTUM 4386/4885ALDH1A1 380/4885NPSR1 582/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.