SCHEMBL3462992

SCHEMBL3462992

CC(C)NCC(O)COc1ccc(CCO)cc1

nearest known ligand 0.77

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 5/20 0.75
ADRB1 P08588 4/20 0.75
CYP2D6 P10635 2/20 0.75
ADRA1A P35348 2/20 0.75
NR3C1 P04150 1/20 0.75
CYP2J2 P51589 1/20 0.75
PDE4D Q08499 1/20 0.75
PTGS1 P23219 1/20 0.68
SLC6A2 P23975 1/20 0.68
ADRB3 P13945 1/20 0.66
ABCB1 P08183 1/20 0.65
LMNA P02545 2/20 0.65
TDP1 Q9NUW8 2/20 0.65
CNR1 P21554 1/20 0.65
ADRA1D P25100 1/20 0.65
ADRA1B P35368 1/20 0.65
KDM4E B2RXH2 1/20 0.65
CYP1A2 P05177 1/20 0.65
GLA P06280 1/20 0.65
CYP3A4 P08684 1/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15159029 0.93 ADRB2 (0.73) ADRB2ADRB1CYP2D6ADRA1ANR3C1
SCHEMBL13204479 0.88 ADRB2 (0.75) ADRB2ADRB1CYP2D6ADRA1ANR3C1
SCHEMBL16341905 0.88 PTGS1 (0.72) ADRB2ADRB1CYP2D6ADRA1ANR3C1
SCHEMBL2585653 0.88 PTGS1 (0.72) ADRB2ADRB1CYP2D6ADRA1ANR3C1
SCHEMBL11651404 0.87 ADRB2 (0.73) ADRB2ADRB1CYP2D6ADRA1ANR3C1
SCHEMBL9452302 0.87 ADRB2 (0.73) ADRB2ADRB1CYP2D6ADRA1ANR3C1
SCHEMBL28412321 0.86 PTGS1 (0.74) ADRB2ADRB1CYP2D6ADRA1ANR3C1
SCHEMBL220354 0.86 ADRB1 (0.76) ADRB2ADRB1CYP2D6ADRA1ANR3C1
Metoprolol SCHEMBL1561123 0.86 ADRB1 (1.00) ADRB2ADRB1CYP2D6ADRA1ANR3C1
(R)-Metoprolol SCHEMBL40918 0.86 ADRB1 (1.00) ADRB2ADRB1CYP2D6ADRA1ANR3C1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111110854-A Composition comprising a histamine release-promoting substance and an inhibitory compound 黄泳华 2020-05-08 CN claimed
CN-111110854-A Composition comprising a histamine release-promoting substance and an inhibitory compound 黄泳华 2020-05-08 CN disclosed
WO-2010029566-A2 PROCESS FOR PREPARATION OF PHENOXYPROPANOL AMINES INDOCO REMEDIES LIMITED (IN) 2010-03-18 WO disclosed
WO-2010029566-A2 PROCESS FOR PREPARATION OF PHENOXYPROPANOL AMINES INDOCO REMEDIES LIMITED (IN) 2010-03-18 WO disclosed
US-4760182-A Process for preparing substituted phenol ethers via oxazolidine-structure intermediates TORCAN CHEMICAL LTD. (CA) 1988-07-26 US disclosed