SCHEMBL22045587

SCHEMBL22045587

c1cc2cnncc2c2cnncc12

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.34
ALDH1A1 P00352 3/20 0.34
TP53 P04637 2/20 0.34
CYP3A4 P08684 2/20 0.34
GOT1 P17174 2/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
NPC1 O15118 1/20 0.34
LMNA P02545 1/20 0.34
MPO P05164 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2D6 P10635 1/20 0.34
PKM P14618 1/20 0.34
MAOA P21397 1/20 0.34
PTGS1 P23219 1/20 0.34
THPO P40225 1/20 0.34
RAB9A P51151 1/20 0.34
AOX1 Q06278 1/20 0.34
ACOX1 Q15067 1/20 0.34
TDP1 Q9NUW8 2/20 0.33
MAPT P10636 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2407872 0.84 ALDH1A1 (0.60) KDM4EALDH1A1TP53CYP3A4GOT1
SCHEMBL29350993 0.84 ALDH1A1 (0.60) KDM4EALDH1A1TP53CYP3A4GOT1
SCHEMBL18099780 0.82 CLK1 (0.46) KDM4ECYP3A4LMNACYP1A2CYP2D6
SCHEMBL18099790 0.82 IMPDH2 (0.48) KDM4EALDH1A1CYP3A4LMNACYP1A2
SCHEMBL22045540 0.80 HPRT1 (0.64) KDM4EALDH1A1TP53CYP3A4GOT1
SCHEMBL8404449 0.78 TSHR (0.50) KDM4EALDH1A1CYP3A4LMNACYP1A2
SCHEMBL22044866 0.76 PKM (0.38) CYP3A4PKMGPR3
SCHEMBL9618221 0.76 CYP2A6 (0.48) CYP3A4CYP1A2MAOAIMPDH2CYP2A6
SCHEMBL30539248 0.73 CLK1 (0.33) KDM4E
SCHEMBL22045622 0.72 CLK1 (0.39) KDM4ETP53CYP3A4SMN1; SMN2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3052506-B1 AZABORININE DERIVATIVES, THEIR SYNTHESIS AND USE IN ORGANIC ELECTRONIC DEVICES FLEXENABLE LTD (GB) 2020-06-03 EP disclosed