SCHEMBL22046331

SCHEMBL22046331

CS(=O)(=O)c1cc(N)ccc1C#N

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.52
KDM4E B2RXH2 8/20 0.49
ALDH1A1 P00352 4/20 0.49
USP2 O75604 1/20 0.49
HTT P42858 1/20 0.40
LMNA P02545 2/20 0.39
KCNJ1 P48048 1/20 0.38
KCNH2 Q12809 1/20 0.38
HPGD P15428 3/20 0.37
MAPT P10636 2/20 0.37
CYP3A4 P08684 2/20 0.36
CYP2D6 P10635 2/20 0.36
CYP2C19 P33261 2/20 0.36
CYP2C9 P11712 1/20 0.36
NR1H2 P55055 1/20 0.36
NR1H3 Q13133 1/20 0.36
MEN1 O00255 1/20 0.35
CYP1A2 P05177 1/20 0.35
KMT2A Q03164 1/20 0.35
SLC22A12 Q96S37 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29452111 0.81 ALDH1A1 (0.60) L3MBTL1KDM4EALDH1A1USP2HTT
SCHEMBL12327903 0.79 SGK1 (0.41) KDM4EALDH1A1HTTKCNJ1KCNH2
SCHEMBL10164103 0.79 RAD51 (0.45) ALDH1A1HTTKCNJ1KCNH2NR1H2
SCHEMBL12560129 0.78 VCAM1 (0.46) ALDH1A1HTTMEN1KMT2ASLC22A12
SCHEMBL21013691 0.78 ALDH1A1 (0.40) ALDH1A1HTTKCNJ1KCNH2NR1H2
SCHEMBL1271815 0.78 EPAS1 (0.42) ALDH1A1HTTKCNJ1KCNH2MEN1
SCHEMBL17505017 0.78 MAOB (0.40) KDM4EALDH1A1USP2HTTLMNA
SCHEMBL15545328 0.77 ALDH1A1 (0.41) KDM4EALDH1A1USP2LMNAHPGD
SCHEMBL19742421 0.75 KDM4E (0.46) L3MBTL1KDM4EALDH1A1USP2LMNA
SCHEMBL9175606 0.74 L3MBTL1 (0.61) L3MBTL1KDM4EALDH1A1USP2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2970252-B1 SUBSTITUTED 2-AZA-BICYCLO[2.2.2]OCTANE-3-CARBOXYLIC ACID (BENZYL-CYANO-METHYL)-AMIDES INHIBITORS OF CATHEPSIN C BOEHRINGER INGELHEIM INT (DE) 2020-06-03 EP disclosed