SCHEMBL22047604

SCHEMBL22047604

COc1c(C(C)=O)cc(Cl)c(C)c1N1CCCC1O

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 7/20 0.40
CYP1A2 P05177 2/20 0.35
CYP2D6 P10635 2/20 0.35
DRD4 P21917 2/20 0.35
DRD3 P35462 2/20 0.35
KMT2A Q03164 2/20 0.35
KDM4E B2RXH2 1/20 0.35
CYP2C9 P11712 1/20 0.35
DRD1 P21728 1/20 0.35
DRD5 P21918 1/20 0.35
CYP2C19 P33261 1/20 0.35
HSD17B10 Q99714 1/20 0.35
MEN1 O00255 1/20 0.34
LMNA P02545 1/20 0.34
HIF1A Q16665 1/20 0.34
ACHE P22303 1/20 0.34
HTR4 Q13639 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9929042 0.81 DRD2 (0.36) DRD2ACHEHTR4
SCHEMBL9970971 0.77 HPGD (0.32)
SCHEMBL9928921 0.76 ATM (0.42) KMT2AMEN1LMNA
SCHEMBL9970967 0.74 HCRTR1 (0.35)
SCHEMBL14753934 0.72 IMPDH2 (0.48) KDM4EHSD17B10
SCHEMBL14736962 0.70 ALDH1A1 (0.37) DRD2KMT2AHSD17B10MEN1LMNA
SCHEMBL9928890 0.69 IMPDH2 (0.34) DRD2HSD17B10LMNA
SCHEMBL14742470 0.69 PIK3CD (0.35) DRD2CYP1A2CYP2D6DRD4DRD3
SCHEMBL9929296 0.68 HSD17B10 (0.40) KDM4EHSD17B10
SCHEMBL9928807 0.68 IMPDH2 (0.39) KMT2AKDM4EHSD17B10MEN1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3660016-A1 N-(1-(SUBSTITUTED-PHENYL)ETHYL)-9H-PURIN-6-AMINES AS PI3K INHIBITORS Incyte Holdings Corporation (US) 2020-06-03 EP disclosed