SCHEMBL22064142

SCHEMBL22064142

COC(=O)CCCCC(=O)NC(C(=O)NCC(=O)OC(C)(C)C)C(C)C

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CTSS P25774 2/20 0.45
CTSK P43235 2/20 0.45
RECQL P46063 1/20 0.44
FURIN P09958 1/20 0.38
CAPN1 P07384 1/20 0.36
TSHR P16473 1/20 0.36
CA2 P00918 2/20 0.35
CA1 P00915 1/20 0.35
CA7 P43166 1/20 0.35
CYP2D6 P10635 1/20 0.35
BIRC2 Q13490 1/20 0.35
SDCBP O00560 1/20 0.35
SDC2 P34741 1/20 0.35
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35
KLK5 Q9Y337 1/20 0.34
GAA P10253 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22064353 0.87 CTSS (0.43) CTSSCTSKRECQLFURINCAPN1
SCHEMBL22987335 0.86 RECQL (0.46) RECQLCAPN1TSHRBIRC2ALDH1A1
SCHEMBL19656347 0.83 PSENEN (0.40) CTSSCTSKRECQLTSHRCA2
SCHEMBL25908085 0.83 PSENEN (0.40) CTSSCTSKRECQLTSHRCA2
SCHEMBL464264 0.80 CTSS (0.43) CTSSCTSKCA2CA1CA7
SCHEMBL19471807 0.80 RECQL (0.69) RECQLTSHRCA2ALDH1A1LMNA
SCHEMBL22508225 0.78 RECQL (0.39) RECQLTSHRALDH1A1LMNA
SCHEMBL4470428 0.77 CTSK (0.67) CTSSCTSKCA2CA1CA7
SCHEMBL9788528 0.77 CTSK (0.67) CTSSCTSKCA2CA1CA7
SCHEMBL22960908 0.77 CTSK (0.59) CTSSCTSKCAPN1CA2CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3778601-A1 CYTOTOXIC BENZODIAZEPINE DERIVATIVES ImmunoGen, Inc. (US) 2021-02-17 EP disclosed
EP-3189056-B1 CYTOTOXIC BENZODIAZEPINE DERIVATIVES IMMUNOGEN INC (US) 2020-06-10 EP disclosed