SCHEMBL22065355

SCHEMBL22065355

CNc1nc(-c2cccc(Cl)c2)nc(Nc2cc(C(=O)Nc3cccc(C(F)(F)F)c3)ccc2C)c1C=N

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LCK P06239 6/20 0.54
MAPK14 Q16539 5/20 0.54
BRAF P15056 5/20 0.54
SRC P12931 3/20 0.54
EPHB2 P29323 3/20 0.54
DDR1 Q08345 3/20 0.54
DDR2 Q16832 3/20 0.54
LMNA P02545 3/20 0.54
KDR P35968 3/20 0.54
ESYT2 A0FGR8 2/20 0.54
NBAS A2RRP1 2/20 0.54
CNOT1 A5YKK6 2/20 0.54
TBKBP1 A7MCY6 2/20 0.54
AGPS O00116 2/20 0.54
MYO1F O00160 2/20 0.54
SNAP23 O00161 2/20 0.54
AP3B1 O00203 2/20 0.54
PSMD12 O00232 2/20 0.54
BMPR1B O00238 2/20 0.54
PGRMC1 O00264 2/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22066412 0.92 POLB (0.57) LCKMAPK14BRAFSRCEPHB2
SCHEMBL22066322 0.92 LCK (0.54) LCKMAPK14BRAFSRCEPHB2
SCHEMBL22065360 0.89 POLB (0.53) LCKMAPK14BRAFSRCEPHB2
SCHEMBL22066328 0.86 POLB (0.55) LCKMAPK14BRAFSRCEPHB2
SCHEMBL22066074 0.82 BRAF (0.61) LCKMAPK14BRAFSRCEPHB2
SCHEMBL22025325 0.81 POLB (0.56) LCKMAPK14BRAFSRCEPHB2
SCHEMBL22066484 0.80 MAPK14 (0.68) LCKMAPK14BRAFSRCEPHB2
SCHEMBL22024561 0.80 BRAF (0.81) LCKMAPK14BRAFSRCEPHB2
SCHEMBL21975658 0.76 KDR (0.57) LCKMAPK14BRAFSRCEPHB2
SCHEMBL22024546 0.76 PIKFYVE (0.71) LCKMAPK14BRAFSRCEPHB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3663293-A1 SUBSTITUTED PENTA- AND HEXA-HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, DRUG COMBINATION AND USE THEREOF Xiamen University (CN) 2020-06-10 EP disclosed