SCHEMBL22069710

SCHEMBL22069710

CC(C)c1ccc(Oc2ccc(N)cc2Cl)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE7A Q13946 2/20 0.54
FFAR1 O14842 2/20 0.48
NPBWR1 P48145 1/20 0.45
MCHR1 Q99705 1/20 0.45
HTR2A P28223 1/20 0.44
SLC6A4 P31645 1/20 0.44
MAOA P21397 1/20 0.44
MAOB P27338 1/20 0.44
PNLIP P16233 1/20 0.42
ALDH1A1 P00352 6/20 0.42
CYP3A4 P08684 3/20 0.42
TSHR P16473 2/20 0.42
TDP1 Q9NUW8 2/20 0.42
SMN1; SMN2 Q16637 3/20 0.42
HTR2C P28335 1/20 0.41
HTR2B P41595 1/20 0.41
MAPT P10636 4/20 0.41
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
KDM4E B2RXH2 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4318630 0.89 PDE7A (0.63) PDE7AHTR2ASLC6A4MAOAMAOB
SCHEMBL2509239 0.89 PDE7A (0.56) PDE7AFFAR1NPBWR1MCHR1HTR2A
SCHEMBL22452604 0.85 PDE7A (0.52) PDE7AFFAR1NPBWR1MCHR1HTR2A
SCHEMBL21925217 0.85 MAPT (0.50) PDE7ANPBWR1MCHR1MAOAMAOB
SCHEMBL22966319 0.83 ALDH1A1 (0.46) PDE7AFFAR1NPBWR1MCHR1HTR2A
SCHEMBL5583563 0.83 TEAD4 (0.57) PDE7AHTR2ASLC6A4MAOAMAOB
SCHEMBL21620367 0.83 FFAR1 (0.65) FFAR1HTR2ASLC6A4ALDH1A1TDP1
SCHEMBL1147436 0.83 PDE7A (0.53) PDE7AHTR2ASLC6A4MAOAMAOB
SCHEMBL8904604 0.82 PDE7A (0.59) PDE7AHTR2ASLC6A4MAOAMAOB
SCHEMBL554722 0.82 MAOA (0.61) PDE7AFFAR1HTR2ASLC6A4MAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3666769-A1 NOVEL CASPASE INHIBITORS RIJKSUNIVERSITEIT GRONINGEN (NL) 2020-06-17 EP disclosed
EP-3666769-A1 NOVEL CASPASE INHIBITORS RIJKSUNIVERSITEIT GRONINGEN (NL) 2020-06-17 EP disclosed