SCHEMBL22071810

SCHEMBL22071810

CCSc1nc2c(cnn2C2CCSCC2)c(=O)[nH]1

nearest known ligand 0.52

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.52
ESR1 P03372 1/20 0.52
L3MBTL1 Q9Y468 1/20 0.52
PDE9A O76083 16/20 0.49
SMN1; SMN2 Q16637 1/20 0.46
PDE1C Q14123 1/20 0.45
PDE1B Q01064 1/20 0.43
ALDH1A1 P00352 1/20 0.43
TSHR P16473 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22072396 0.92 LMNA (0.57) LMNAESR1L3MBTL1PDE9ASMN1; SMN2
SCHEMBL22072398 0.88 PDE9A (0.61) LMNAESR1L3MBTL1PDE9APDE1C
SCHEMBL22072367 0.87 PDE9A (0.46) PDE9APDE1CPDE1B
SCHEMBL22072364 0.86 PDE9A (0.47) ESR1PDE9APDE1CPDE1BALDH1A1
SCHEMBL22072366 0.85 CYP1A2 (0.59) L3MBTL1PDE9ASMN1; SMN2ALDH1A1TSHR
SCHEMBL22071807 0.84 PDE9A (0.56) LMNAESR1L3MBTL1PDE9A
SCHEMBL22042934 0.82 SMN1; SMN2 (0.47) LMNASMN1; SMN2ALDH1A1TSHR
SCHEMBL22042861 0.78 PDE9A (0.50) PDE9APDE1CPDE1B
SCHEMBL22042836 0.77 ALDH1A1 (0.50) ESR1PDE9APDE1CPDE1BALDH1A1
SCHEMBL7879153 0.77 PDE9A (0.74) PDE9APDE1C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020116972-A1 COMPOUNDS HAVING PDE9A INHIBITORY ACTIVITY, AND PHARMACEUTICAL USES THEREOF 한국화학연구원 2020-06-11 WO disclosed