SCHEMBL22072044

SCHEMBL22072044

OC[C@@H]1CNCCN1c1nc(Nc2cc(-c3ccccc3)[nH]n2)c2ccccc2n1

nearest known ligand 0.56

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SPAST Q9UBP0 1/20 0.56
PAK4 O96013 3/20 0.51
NTRK1 P04629 2/20 0.48
PAK1 Q13153 2/20 0.45
AURKA O14965 2/20 0.42
FLT1 P17948 1/20 0.42
KDR P35968 1/20 0.42
FLT3 P36888 1/20 0.42
HTR2A P28223 5/20 0.41
SRC P12931 2/20 0.41
GSK3B P49841 2/20 0.41
EIF2AK2 P19525 1/20 0.41
GSK3A P49840 1/20 0.41
AURKB Q96GD4 1/20 0.41
CHEK1 O14757 1/20 0.40
CCNA2 P20248 1/20 0.39
CDK2 P24941 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22072040 0.91 SPAST (0.59) SPASTPAK4NTRK1PAK1AURKA
SCHEMBL22072048 0.86 SPAST (0.77) SPASTPAK4PAK1AURKAHTR2A
SCHEMBL22072526 0.79 SPAST (0.67) SPASTPAK4NTRK1PAK1AURKA
SCHEMBL22072735 0.77 SPAST (0.67) SPASTPAK4NTRK1PAK1AURKA
SCHEMBL20352282 0.76 PAK4 (0.60) PAK4NTRK1PAK1AURKAAURKB
SCHEMBL22072525 0.75 HRH4 (0.63) PAK4NTRK1PAK1AURKAFLT1
SCHEMBL22072085 0.74 PAK4 (0.66) PAK4NTRK1PAK1SRCGSK3B
SCHEMBL22072736 0.73 SPAST (0.66) SPASTPAK4PAK1AURKAHTR2A
SCHEMBL22035049 0.72 SPAST (1.00) SPASTPAK4PAK1HTR2A
SCHEMBL22035048 0.72 SPAST (1.00) SPASTPAK4PAK1HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020118183-A1 2,4-DIAMINOPYRIMIDINE BICYCLES FOR TREATING CANCER KAPOOR TARUN M (US) 2020-06-11 WO disclosed