SCHEMBL22072736

SCHEMBL22072736

Cc1cc(C)c(C)c(-c2cc(Nc3nc(N4CCNC[C@H]4C)nc4ccccc34)n[nH]2)c1

nearest known ligand 0.66

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SPAST Q9UBP0 1/20 0.66
PAK4 O96013 7/20 0.46
PAK1 Q13153 4/20 0.46
AURKA O14965 5/20 0.38
SRC P12931 3/20 0.38
GSK3B P49841 3/20 0.38
AURKB Q96GD4 3/20 0.38
EIF2AK2 P19525 1/20 0.38
GSK3A P49840 1/20 0.38
HTR2A P28223 3/20 0.38
ROCK2 O75116 1/20 0.38
ROCK1 Q13464 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22072526 0.81 SPAST (0.67) SPASTPAK4PAK1AURKASRC
SCHEMBL22072735 0.81 SPAST (0.67) SPASTPAK4PAK1AURKASRC
SCHEMBL22035049 0.80 SPAST (1.00) SPASTPAK4PAK1HTR2A
SCHEMBL22035048 0.80 SPAST (1.00) SPASTPAK4PAK1HTR2A
SCHEMBL22072081 0.77 SPAST (0.72) SPASTPAK4PAK1AURKAAURKB
SCHEMBL22072040 0.75 SPAST (0.59) SPASTPAK4PAK1AURKASRC
SCHEMBL22072044 0.73 SPAST (0.56) SPASTPAK4PAK1AURKASRC
SCHEMBL22072048 0.68 SPAST (0.77) SPASTPAK4PAK1AURKAAURKB
SCHEMBL22072740 0.68 SPAST (0.76) SPASTPAK4PAK1AURKAAURKB
SCHEMBL5787049 0.66 ALDH1A1 (0.64) SPASTROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020118183-A1 2,4-DIAMINOPYRIMIDINE BICYCLES FOR TREATING CANCER KAPOOR TARUN M (US) 2020-06-11 WO disclosed