SCHEMBL22075531

SCHEMBL22075531

C=Nc1ncnc2[nH]nc(-c3ccc(OC)c(F)c3)c12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.40
KDM4E B2RXH2 2/20 0.40
MAPK1 P28482 1/20 0.40
KIT P10721 6/20 0.39
CDK2 P24941 1/20 0.38
MEN1 O00255 1/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
KMT2A Q03164 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
PTGS1 P23219 1/20 0.38
PTGS2 P35354 1/20 0.38
PDGFRB P09619 1/20 0.37
PDGFRA P16234 1/20 0.37
RAF1 P04049 1/20 0.37
BRAF P15056 1/20 0.37
CSF1R P07333 1/20 0.36
JAK2 O60674 1/20 0.35
JAK3 P52333 1/20 0.35
CYP17A1 P05093 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11306 0.83 SRC (0.47) ALDH1A1KDM4EMAPK1KITMEN1
SCHEMBL10811 0.74 SRC (0.57) KITPIK3CDABL1EGFRHCK
SCHEMBL217790 0.72 ABL1 (0.49) PIK3CDABL1EGFRHCKSRC
SCHEMBL149180 0.72 PIK3CD (0.55) ALDH1A1KDM4EPIK3CDABL1EGFR
SCHEMBL13717800 0.71 CSNK1E (0.45) PIK3CDABL1EGFRHCKSRC
SCHEMBL13717774 0.70 PIK3CD (0.41) KITPIK3CDABL1EGFRHCK
SCHEMBL13718435 0.70 MKNK1 (0.39) PIK3CDEGFRPIK3CG
SCHEMBL19414295 0.69 SRC (0.47) PIK3CDABL1EGFRHCKSRC
SCHEMBL13717565 0.69 LRRK2 (0.40) CSF1RPIK3CDPIK3CG
SCHEMBL22692856 0.68 ERBB2 (0.50) PIK3CDSRCPIK3CAPIK3CBPIK3CG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020113642-A1 SELECTIVE PI3Kδ INHIBITOR AND USE THEREOF 安徽中科拓苒药物科学研究有限公司 2020-06-11 WO disclosed