SCHEMBL22101400

SCHEMBL22101400

Bc1cc(F)c2nc(CC)cc(=O)n2c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CXCR2 P25025 2/20 0.38
KDM5B Q9UGL1 1/20 0.37
MAT2A P31153 1/20 0.36
MAPT P10636 3/20 0.34
POLB P06746 2/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
GRIN1 Q05586 2/20 0.33
GRIN2A Q12879 2/20 0.33
TSHR P16473 2/20 0.33
HSD17B10 Q99714 2/20 0.33
HTT P42858 1/20 0.33
GRIA2 P42262 1/20 0.32
HPGD P15428 2/20 0.32
PKM P14618 2/20 0.32
KDM4E B2RXH2 2/20 0.32
ALDH1A1 P00352 2/20 0.32
TP53 P04637 1/20 0.31
THRB P10828 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22101725 0.85 GRIN1 (0.40) CXCR2KDM5BMAT2AMAPTPOLB
SCHEMBL22393919 0.84 KDM5B (0.36) CXCR2KDM5BMAT2AMAPTPOLB
SCHEMBL22101411 0.84 KDM5B (0.36) CXCR2KDM5BMAT2AMAPTPOLB
SCHEMBL22393704 0.81 MAPT (0.36) CXCR2KDM5BMAT2AMAPTPOLB
SCHEMBL22101447 0.73 BCAT2 (0.33) CXCR2MAT2ABCAT2BCAT1
SCHEMBL22101360 0.73 MAPT (0.35) CXCR2MAT2AMAPTPOLBTP53
SCHEMBL22101696 0.72 KDM5B (0.39) KDM5BMAT2AMAPTPOLBL3MBTL1
SCHEMBL22101695 0.70 MAPT (0.40) KDM5BMAT2AMAPTPOLBL3MBTL1
SCHEMBL22101427 0.70 PABPC1 (0.42) KDM5BMAT2AMAPTL3MBTL1TSHR
SCHEMBL22101884 0.69 MAPT (0.37) KDM5BMAT2AMAPTPOLBL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3666772-A1 DIARYLTHIOHYDANTOIN COMPOUND AS ANDROGEN RECEPTOR ANTAGONIST Chia Tai Tianqing Pharmaceutical Group Co., Ltd. (CN) 2020-06-17 EP disclosed