SCHEMBL22101522

SCHEMBL22101522

Cc1cc(F)c2nc(C(F)F)cc(=O)n2c1

nearest known ligand 0.37

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PIK3CB P42338 17/20 0.37
KCNQ3 O43525 1/20 0.35
KCNQ2 O43526 1/20 0.35
RAD51 Q06609 1/20 0.35
PIK3CD O00329 12/20 0.34
PIK3CA P42336 11/20 0.34
PIK3R1 P27986 1/20 0.33
CSNK1A1 P48729 1/20 0.33
PIK3CG P48736 1/20 0.33
PTK2 Q05397 1/20 0.33
CLK4 Q9HAZ1 1/20 0.33
TDP1 Q9NUW8 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22101697 0.82 KCNQ3 (0.34) PIK3CBKCNQ3KCNQ2RAD51
SCHEMBL22101454 0.82 KCNQ3 (0.35) KCNQ3KCNQ2RAD51
SCHEMBL22101486 0.82 KCNQ3 (0.35) KCNQ3KCNQ2RAD51
SCHEMBL22393588 0.81 KCNQ3 (0.36) KCNQ3KCNQ2RAD51
SCHEMBL22101540 0.76 CYP2C9 (0.35) PIK3CBPIK3CDPIK3CA
SCHEMBL22101725 0.76 GRIN1 (0.40) TDP1L3MBTL1
SCHEMBL22101865 0.73 KCNQ3 (0.31) PIK3CBKCNQ3KCNQ2RAD51
SCHEMBL22101541 0.72 MAPT (0.35) PIK3CB
SCHEMBL22101539 0.70 FFAR4 (0.35) PIK3CB
SCHEMBL25818875 0.70 PDE10A (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3666772-A1 DIARYLTHIOHYDANTOIN COMPOUND AS ANDROGEN RECEPTOR ANTAGONIST Chia Tai Tianqing Pharmaceutical Group Co., Ltd. (CN) 2020-06-17 EP disclosed