SCHEMBL22101697

SCHEMBL22101697

CC(C)c1cc(F)c2nc(C(F)F)cc(=O)n2c1

nearest known ligand 0.34

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KCNQ3 O43525 1/20 0.34
KCNQ2 O43526 1/20 0.34
RAD51 Q06609 1/20 0.33
LMNA P02545 1/20 0.30
TP53 P04637 1/20 0.30
HPGD P15428 1/20 0.30
TSHR P16473 1/20 0.30
HTT P42858 1/20 0.30
HSD17B10 Q99714 1/20 0.30
PIK3CB P42338 1/20 0.30
KDM5B Q9UGL1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22101522 0.82 PIK3CB (0.37) KCNQ3KCNQ2RAD51PIK3CB
SCHEMBL22101486 0.79 KCNQ3 (0.35) KCNQ3KCNQ2RAD51
SCHEMBL22101454 0.79 KCNQ3 (0.35) KCNQ3KCNQ2RAD51
SCHEMBL22393588 0.79 KCNQ3 (0.36) KCNQ3KCNQ2RAD51
SCHEMBL22101698 0.76 KDM4E (0.39) TP53HPGDHSD17B10
SCHEMBL22393590 0.76 ELANE (0.32) TSHR
SCHEMBL25105584 0.72 EGFR (0.31)
SCHEMBL22101865 0.71 KCNQ3 (0.31) KCNQ3KCNQ2RAD51PIK3CB
SCHEMBL19836282 0.70 EGFR (0.37)
SCHEMBL22101455 0.70 P2RX3 (0.36) PIK3CB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3666772-A1 DIARYLTHIOHYDANTOIN COMPOUND AS ANDROGEN RECEPTOR ANTAGONIST Chia Tai Tianqing Pharmaceutical Group Co., Ltd. (CN) 2020-06-17 EP disclosed