SCHEMBL22101541

SCHEMBL22101541

CCOc1cc(=O)n2cc(C)cc(F)c2n1

nearest known ligand 0.35

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.35
RXFP1 Q9HBX9 3/20 0.35
KDM4E B2RXH2 2/20 0.35
ALDH1A1 P00352 2/20 0.35
ADORA2A P29274 1/20 0.35
ADORA1 P30542 1/20 0.35
PIK3CB P42338 2/20 0.33
GRIN1 Q05586 1/20 0.33
GRIN2A Q12879 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
POLB P06746 2/20 0.32
LMNA P02545 2/20 0.32
TP53 P04637 1/20 0.32
BCAT2 O15382 1/20 0.32
PDE5A O76074 1/20 0.31
PKM P14618 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22101539 0.85 FFAR4 (0.35) MAPTRXFP1KDM4EALDH1A1PIK3CB
SCHEMBL22101536 0.85 THRB (0.38) MAPTRXFP1KDM4EALDH1A1PIK3CB
SCHEMBL22101868 0.85 KDM4E (0.35) MAPTRXFP1KDM4EADORA2AADORA1
SCHEMBL22101540 0.84 CYP2C9 (0.35) RXFP1KDM4EALDH1A1PIK3CBGRIN1
SCHEMBL24425379 0.83 MAPT (0.34) MAPTALDH1A1ADORA2AADORA1TP53
SCHEMBL22393590 0.83 ELANE (0.32) ADORA2AADORA1
SCHEMBL22101725 0.78 GRIN1 (0.40) MAPTRXFP1KDM4EALDH1A1GRIN1
SCHEMBL22101452 0.75 MAPT (0.33) MAPTPIK3CBPDE5A
SCHEMBL22101522 0.72 PIK3CB (0.37) PIK3CB
SCHEMBL22101709 0.71 GRIN1 (0.32) RXFP1KDM4EALDH1A1GRIN1GRIN2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3666772-A1 DIARYLTHIOHYDANTOIN COMPOUND AS ANDROGEN RECEPTOR ANTAGONIST Chia Tai Tianqing Pharmaceutical Group Co., Ltd. (CN) 2020-06-17 EP disclosed