SCHEMBL22110461

SCHEMBL22110461

Brc1cc(Br)cc(CI)c1

nearest known ligand 0.44

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.44
TAAR1 Q96RJ0 1/20 0.31
CYP3A4 P08684 1/20 0.30
TSHR P16473 1/20 0.30
TDP1 Q9NUW8 1/20 0.30
AGXT P21549 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8447346 0.84 IDO1 (0.33) IDO1TSHR
SCHEMBL28056120 0.82 TACR1 (0.40) IDO1
SCHEMBL7596361 0.77 ALDH1A1 (0.43) IDO1TAAR1
SCHEMBL17994035 0.77 NOTUM (0.40) IDO1TAAR1
SCHEMBL5442950 0.75 ALDH1A1 (0.30)
SCHEMBL3070777 0.75 POLB (0.42) TSHRTDP1
SCHEMBL1044848 0.75 IDO1 (0.44) IDO1TAAR1CYP3A4TSHRTDP1
SCHEMBL1542275 0.73 IDO1 (0.48) IDO1TAAR1CYP3A4TSHRTDP1
SCHEMBL2197501 0.73
SCHEMBL7600112 0.73 IDO1 (0.38) IDO1TAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2825536-B1 BIS-QUARTERNARY CINCHONA ALKALOID SALTS AS ASYMMETRIC PHASE TRANSFER CATALYSTS MERCK SHARP & DOHME (US) 2020-06-17 EP disclosed