SCHEMBL22114122

SCHEMBL22114122

COc1cc(OC)cc(Oc2ccc(C)cc2F)c1

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ACHE P22303 3/20 0.45
ALDH1A1 P00352 2/20 0.41
CYP3A4 P08684 1/20 0.41
NQO2 P16083 1/20 0.41
TRPA1 O75762 2/20 0.38
AR P10275 3/20 0.38
MAPK14 Q16539 1/20 0.38
HTR1A P08908 1/20 0.38
SLC6A2 P23975 1/20 0.38
SLC6A4 P31645 1/20 0.38
RELA Q04206 1/20 0.37
NPC1 O15118 1/20 0.37
MAPT P10636 1/20 0.37
RAB9A P51151 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
TUBB1 Q9H4B7 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22199016 0.89 ACHE (0.50) ACHEALDH1A1CYP3A4TRPA1AR
SCHEMBL779089 0.88 ACHE (0.53) ACHEALDH1A1ARMAPK14SLC6A2
SCHEMBL27115327 0.85 ALDH1A1 (0.44) ACHEALDH1A1CYP3A4HTR1ASLC6A2
SCHEMBL14662668 0.83 EPAS1 (0.42) ACHEHTR1ASLC6A2SLC6A4
SCHEMBL26186321 0.83 SLC6A4 (0.39) ACHEALDH1A1CYP3A4TRPA1HTR1A
SCHEMBL22199022 0.82 HSPB1 (0.45) ACHEALDH1A1ARHTR1ASLC6A2
SCHEMBL26493853 0.82 ACHE (0.46) ACHEALDH1A1CYP3A4TRPA1HTR1A
SCHEMBL22069740 0.80 CYP19A1 (0.43) ALDH1A1CYP3A4NQO2TRPA1MAPT
SCHEMBL27115328 0.80 EPAS1 (0.38) ACHEALDH1A1HTR1ASLC6A2SLC6A4
SCHEMBL11883 0.80 ACHE (0.62) ACHEALDH1A1CYP3A4NPC1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3666769-A1 NOVEL CASPASE INHIBITORS RIJKSUNIVERSITEIT GRONINGEN (NL) 2020-06-17 EP disclosed