SCHEMBL2211558

SCHEMBL2211558

N#CC(C(=O)Cl)c1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.48
TRPA1 O75762 1/20 0.43
TDP1 Q9NUW8 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
CYP2D6 P10635 1/20 0.41
SRC P12931 1/20 0.41
LMNA P02545 5/20 0.41
ALDH1A1 P00352 3/20 0.41
USP2 O75604 1/20 0.41
HPGD P15428 1/20 0.41
HTT P42858 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
AKR1C3 P42330 1/20 0.41
AKR1C1 Q04828 1/20 0.41
HDAC3 O15379 1/20 0.41
HDAC4 P56524 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC7 Q8WUI4 1/20 0.41
HDAC2 Q92769 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11813692 0.83 TSHR (0.52) TSHRTRPA1TDP1L3MBTL1CYP2D6
SCHEMBL1019171 0.83 TSHR (0.52) TSHRTRPA1TDP1L3MBTL1CYP2D6
Ammonia Solution, Strong SCHEMBL38661532 0.81 TSHR (0.50) TSHRTRPA1TDP1L3MBTL1CYP2D6
SCHEMBL6960576 0.81 TSHR (0.50) TSHRTRPA1TDP1L3MBTL1CYP2D6
SCHEMBL10432296 0.79 TSHR (0.48) TSHRTRPA1TDP1L3MBTL1CYP2D6
SCHEMBL2927032 0.79 TSHR (0.48) TSHRTRPA1TDP1L3MBTL1CYP2D6
SCHEMBL2771881 0.79 TSHR (0.48) TSHRTRPA1TDP1L3MBTL1CYP2D6
SCHEMBL1720075 0.79 ALDH1A1 (0.49) TSHRTRPA1TDP1L3MBTL1CYP2D6
SCHEMBL10439400 0.79 LMNA (0.44) TSHRTRPA1TDP1L3MBTL1CYP2D6
SCHEMBL5505530 0.78 L3MBTL1 (0.61) TSHRTRPA1TDP1L3MBTL1CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2348120-B1 Enzymatic reduction of 1-phenylpropanone and derivatives thereof Universität Wien (AT) 2014-06-11 EP disclosed
EP-2348120-A1 Enzymatic reduction of 1-phenylpropanone and derivatives thereof Universität Wien (AT) 2011-07-27 EP disclosed
US-4005074-A Process for cleaving an imido side chain from penicillins and cephalosporins ELI LILLY AND COMPANY (US) 1977-01-25 US disclosed
US-4001239-A CEPHALOSPORIN CLEAVAGE PROCESS ELI LILLY AND COMPANY (US) 1977-01-04 US disclosed
US-3994888-A Cephalosporin cleavage process ELI LILLY AND COMPANY (US) 1976-11-30 US disclosed