SCHEMBL2213569

SCHEMBL2213569

COC(=O)C(C1CCN(C(=O)O)C(C(C)(C)C)C1)C(O)c1ccc(F)cc1NC(=O)C(C)(C)C

nearest known ligand 0.34

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
NR3C2 P08235 1/20 0.34
CHRM3 P20309 6/20 0.32
NTRK1 P04629 1/20 0.32
KCNT1 Q5JUK3 1/20 0.31
GAA P10253 1/20 0.31
CHRM2 P08172 1/20 0.31
CHRM1 P11229 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2211378 0.84
SCHEMBL5592013 0.83 NR3C2 (0.34) NR3C2CHRM3NTRK1KCNT1GAA
SCHEMBL2213566 0.80 GPR119 (0.45)
SCHEMBL5182812 0.73 DPP4 (0.37)
SCHEMBL4053813 0.72 MAPT (0.37) KCNT1GAA
SCHEMBL2359872 0.70 TSHR (0.34) GAA
SCHEMBL2980219 0.70 ALDH1A1 (0.36) CHRM3
SCHEMBL2212500 0.70 STS (0.41)
SCHEMBL2213653 0.69 DPP4 (0.46)
SCHEMBL2214131 0.66 ALDH1A1 (0.42) CHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2013213-B1 CONSTRAINED COMPOUNDS AS CGRP-RECEPTOR ANTAGONISTS BRISTOL MYERS SQUIBB CO (US) 2011-07-27 EP disclosed