SCHEMBL5592013

SCHEMBL5592013

COC(=O)C(C1CCN(C(C)(C)C)CC1)C(O)c1ccc(F)cc1NC(=O)C(C)(C)C

nearest known ligand 0.34

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
NR3C2 P08235 1/20 0.34
NTRK1 P04629 1/20 0.34
CHRM3 P20309 14/20 0.34
KCNT1 Q5JUK3 1/20 0.33
NPY2R P49146 1/20 0.32
GAA P10253 1/20 0.32
RAB9A P51151 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4053813 0.89 MAPT (0.37) KCNT1GAARAB9A
SCHEMBL2213566 0.87 GPR119 (0.45) RAB9A
SCHEMBL2213569 0.83 NR3C2 (0.34) NR3C2NTRK1CHRM3KCNT1GAA
SCHEMBL4049258 0.82
SCHEMBL5591928 0.81 CHRM3 (0.35) CHRM3RAB9A
SCHEMBL2212500 0.76 STS (0.41) RAB9A
SCHEMBL2213653 0.76 DPP4 (0.46) RAB9A
SCHEMBL2359872 0.70 TSHR (0.34) GAARAB9A
SCHEMBL2980219 0.70 ALDH1A1 (0.36) CHRM3NPY2R
SCHEMBL2211375 0.70 GPR119 (0.40) RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007130860-A2 CONSTRAINED COMPOUNDS AS CGRP-RECEPTOR ANTAGONISTS BRISTOL-MYERS SQUIBB COMPANY (US) 2007-11-15 WO disclosed