SCHEMBL2214037

SCHEMBL2214037

CCOc1ccc2c(c1)C1(CCNCC1)OC2=O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.47
AVPR1A P37288 1/20 0.41
ALK Q9UM73 2/20 0.40
HRH3 Q9Y5N1 1/20 0.40
PDK2 Q15119 1/20 0.40
ALDH1A1 P00352 3/20 0.39
KDM4E B2RXH2 3/20 0.39
HPGD P15428 1/20 0.39
OPRM1 P35372 2/20 0.39
OPRD1 P41143 2/20 0.39
OPRK1 P41145 2/20 0.39
MAPT P10636 3/20 0.38
HSD17B10 Q99714 3/20 0.38
ESR2 Q92731 1/20 0.38
LMNA P02545 2/20 0.37
POLB P06746 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
KMT2A Q03164 3/20 0.36
MEN1 O00255 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL736508 0.85 AVPR1A (0.53) AVPR1AHRH3ALDH1A1KDM4EHPGD
SCHEMBL2212850 0.85 PDK2 (0.43) AVPR1AALKHRH3PDK2CA12
Hydrochloric Acid SCHEMBL20955425 0.84 AVPR1A (0.52) AVPR1AHRH3OPRD1KMT2AMEN1
Hydrochloric Acid SCHEMBL6820160 0.79 SIGMAR1 (0.41) AVPR1APDK2ALDH1A1OPRD1MAPT
SCHEMBL3839131 0.75 AVPR1A (0.50) AVPR1ANPY5R
SCHEMBL22057308 0.75 NPY5R (0.45) AVPR1AMAPTNPY5R
SCHEMBL18373156 0.75 NPY5R (0.45) AVPR1AALDH1A1KDM4EOPRM1OPRD1
SCHEMBL4369332 0.75 AKR1A1 (0.41) AVPR1AALKHRH3PDK2CA12
SCHEMBL5136522 0.75 SIGMAR1 (0.42) AVPR1ANPY5R
SCHEMBL736532 0.75 AVPR1A (0.53) AVPR1AHRH3ALDH1A1OPRD1NPY5R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2125726-B1 SPIRO-PIPERIDINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2011-07-27 EP disclosed