SCHEMBL2214210

SCHEMBL2214210

CC(=O)Nc1cccc(-c2ccc(-c3cc4ccnn4c(Nc4ccc(NC(=O)c5ccc6c(c5)CCNC6)cc4)n3)cc2)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
WNT1 P04628 2/20 0.42
GSK3B P49841 2/20 0.42
DYRK1A Q13627 2/20 0.42
F2 P00734 1/20 0.41
PLG P00747 1/20 0.41
PLAU P00749 1/20 0.41
PLAT P00750 1/20 0.41
KLKB1 P03952 1/20 0.41
PRSS1 P07477 1/20 0.41
SLC2A1 P11166 2/20 0.40
MELK Q14680 3/20 0.39
JAK2 O60674 1/20 0.39
POLB P06746 1/20 0.39
MCL1 Q07820 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
ROCK2 O75116 2/20 0.39
CLK2 P49760 1/20 0.39
CLK3 P49761 1/20 0.39
EGFR P00533 1/20 0.38
ERBB2 P04626 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2214775 0.89 PLAU (0.49) WNT1GSK3BDYRK1AF2PLG
SCHEMBL2213856 0.87 MELK (0.48) WNT1GSK3BDYRK1AF2PLG
SCHEMBL2215892 0.87 PLG (0.45) WNT1GSK3BDYRK1AF2PLG
SCHEMBL2211714 0.86 MELK (0.46) WNT1GSK3BDYRK1AF2PLG
SCHEMBL2214893 0.83 PIK3CA (0.40) JAK2POLBMCL1TDP1ROCK2
SCHEMBL2215002 0.82 JAK2 (0.45) JAK2POLBMCL1TDP1MEN1
SCHEMBL2881428 0.81 FYN (0.51) GSK3BPOLBMEN1KMT2ARAD52
SCHEMBL2214475 0.80 JAK2 (0.43) JAK2POLBMCL1TDP1MEN1
SCHEMBL2215111 0.79 F2 (0.40) WNT1GSK3BDYRK1AF2PLG
SCHEMBL2880155 0.79 PLK1 (0.43) JAK2MEN1KMT2ARAD52

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1797096-B1 PYRAZOLOPYRIMIDINES AS INHIBITORS OF PROTEIN KINASE B (AKT) BAYER SCHERING PHARMA AG (DE) 2011-07-27 EP disclosed