SCHEMBL2214751

SCHEMBL2214751

COc1c2ccccc2c(-c2ccc(N(c3ccc(C=C(c4ccccc4)c4ccccc4)cc3)c3ccc(N(c4ccccc4)c4ccccc4)cc3)cc2)c2ccccc12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.39
KDM4E B2RXH2 2/20 0.39
MAPT P10636 2/20 0.39
HPGD P15428 1/20 0.39
PTGS2 P35354 4/20 0.38
MAPK1 P28482 2/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
CYP19A1 P11511 1/20 0.36
CYP11B2 P19099 1/20 0.36
CYP2D6 P10635 1/20 0.36
ESR1 P03372 1/20 0.34
PDE4A P27815 2/20 0.33
PDE4B Q07343 2/20 0.33
PDE4C Q08493 2/20 0.33
PDE4D Q08499 2/20 0.33
RAB9A P51151 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
SLC16A3 O15427 1/20 0.32
SLC16A1 P53985 1/20 0.32
MEN1 O00255 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2085035 0.90 CYP19A1 (0.44) ALDH1A1KDM4EMAPTPTGS2MAPK1
SCHEMBL12774521 0.88 CYP19A1 (0.42) ALDH1A1KDM4EMAPTPTGS2MAPK1
SCHEMBL9971838 0.88 CYP19A1 (0.42) ALDH1A1KDM4EMAPTPTGS2MAPK1
SCHEMBL9971759 0.87 CYP19A1 (0.44) ALDH1A1KDM4EMAPTHPGDPTGS2
SCHEMBL5870391 0.86 LMNA (0.36) ALDH1A1KDM4EHPGDMAPK1SMN1; SMN2
SCHEMBL2213482 0.85 MAPT (0.49) ALDH1A1KDM4EMAPTHPGDPTGS2
SCHEMBL2211757 0.85 PTGS2 (0.41) ALDH1A1KDM4EMAPTPTGS2MAPK1
SCHEMBL2214749 0.84 KDM1A (0.33) ALDH1A1KDM4EMAPTHPGDCYP2D6
SCHEMBL13027920 0.84 CYP19A1 (0.39) ALDH1A1MAPTPTGS2MAPK1CYP19A1
SCHEMBL2213422 0.81 ALOX5 (0.40) ALDH1A1KDM4EMAPTPTGS2MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6989201-B2 Thin film EL device MATSUSHITA ELECTRIC INDUSTRIAL CO., LTD. (JP) 2006-01-24 US claimed
US-20040076854-A1 Thin film EL device MATSUSHITA ELECTRIC INDUSTRIAL CO., LTD. (JP) 2004-04-22 US claimed
US-20030082400-A1 Thin film el device JOLED INC (JP) 2003-05-01 US claimed
EP-1195422-A1 THIN FILM EL DEVICE MATSUSHITA ELECTRIC INDUSTRIAL CO., LTD. (JP) 2002-04-10 EP claimed
EP-1195422-B1 THIN FILM EL DEVICE PANASONIC CORP (JP) 2011-07-27 EP disclosed
US-7083863-B2 Luminous element and method for preparation thereof MATSUSHITA ELECTRIC INDUSTRIAL CO., LTD. (JP) 2006-08-01 US disclosed
US-6989201-B2 Thin film EL device MATSUSHITA ELECTRIC INDUSTRIAL CO., LTD. (JP) 2006-01-24 US disclosed
US-20050194586-A1 Luminous element and method for preparation thereof JOLED INC (JP) 2005-09-08 US disclosed
US-20040076854-A1 Thin film EL device MATSUSHITA ELECTRIC INDUSTRIAL CO., LTD. (JP) 2004-04-22 US disclosed
US-6682832-B2 THIN FILM ELECTROLUMINESCENCE; LOW VOLTAGE EFFICIENCY MATSUSHITA ELECTRIC INDUSTRIAL CO., LTD. (JP) 2004-01-27 US disclosed
US-20030082400-A1 Thin film el device JOLED INC (JP) 2003-05-01 US disclosed
EP-1195422-A1 THIN FILM EL DEVICE MATSUSHITA ELECTRIC INDUSTRIAL CO., LTD. (JP) 2002-04-10 EP disclosed