SCHEMBL2215207

SCHEMBL2215207

COc1cc(F)c(C(=O)O)cc1N

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.50
HTT P42858 3/20 0.46
LMNA P02545 2/20 0.46
MAPK1 P28482 1/20 0.46
RAB9A P51151 1/20 0.46
LCK P06239 1/20 0.44
FYN P06241 1/20 0.44
KDM4E B2RXH2 3/20 0.43
L3MBTL1 Q9Y468 2/20 0.43
HPGD P15428 2/20 0.42
KEAP1 Q14145 1/20 0.42
FABP4 P15090 1/20 0.41
POLB P06746 1/20 0.41
PTGS2 P35354 1/20 0.41
GAA P10253 2/20 0.40
PKM P14618 2/20 0.40
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA3 P07451 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1163576 0.93 ALDH1A1 (0.50) ALDH1A1HTTLMNAMAPK1RAB9A
SCHEMBL29811842 0.93 ALDH1A1 (0.50) ALDH1A1HTTLMNAMAPK1RAB9A
SCHEMBL22222472 0.86 HTT (0.46) ALDH1A1HTTLMNAMAPK1RAB9A
SCHEMBL1766160 0.85 LCK (0.60) ALDH1A1HTTLMNAMAPK1RAB9A
SCHEMBL2902421 0.85 ALDH1A1 (0.56) ALDH1A1HTTLMNALCKFYN
SCHEMBL8901228 0.83 ALDH1A1 (0.59) ALDH1A1HTTLMNALCKFYN
SCHEMBL17700509 0.83 HTT (0.55) ALDH1A1HTTLMNAMAPK1RAB9A
SCHEMBL13596378 0.80 HTT (0.47) ALDH1A1HTTLMNAMAPK1RAB9A
SCHEMBL17774729 0.80 HTT (0.52) ALDH1A1HTTLMNALCKFYN
SCHEMBL28252793 0.80 LMNA (0.50) ALDH1A1HTTLMNAMAPK1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2351731-B1 A GROUP OF AMINO SUBSTITUTED BENZOYL DERIVATIVES AND THEIR PREPARATION AND THEIR USE INST MED BIOTECHNOLOGY CAMS (CN) 2016-02-10 EP disclosed
US-8710098-B2 Group of amino substituted benzoyl derivatives and their preparation and their use Institute of Medicinal Biotechnology Chinese Academy of Medical Science (CN) 2014-04-29 US disclosed
CN-101367749-B A set of mesidino mesitoyl derivant, preparation and application thereof INST MEDICINAL BIOTECHNOLOGY 2013-04-24 CN disclosed
EP-2351731-A1 A GROUP OF AMINO SUBSTITUTED BENZOYL DERIVATIVES AND THEIR PREPARATION AND THEIR USE Institute Of Medicinal Biotechnology, Chinese Academy of Medical Sciences (CN) 2011-08-03 EP disclosed
US-20110178108-A1 Group of amino substituted benzoyl derivatives and their preparation and their use Institute of Medicinal Biotechnology Academy of Medical Science (CN) 2011-07-21 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110178108-A1 Group of amino substituted benzoyl derivatives and their preparation and their use CUL3, APOBEC3G, BRPF3 ALDH1A1 2851/4885HTT 1248/4885LMNA 2812/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.