SCHEMBL1163576

SCHEMBL1163576

COc1cc(C(=O)O)c(F)cc1N

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.50
LCK P06239 1/20 0.49
FYN P06241 1/20 0.49
KDM4E B2RXH2 4/20 0.47
LMNA P02545 2/20 0.46
HTT P42858 2/20 0.46
MAPK1 P28482 1/20 0.46
RAB9A P51151 1/20 0.46
L3MBTL1 Q9Y468 2/20 0.43
HPGD P15428 1/20 0.42
KEAP1 Q14145 1/20 0.42
MYC P01106 1/20 0.41
POLB P06746 2/20 0.41
FABP4 P15090 1/20 0.41
PKM P14618 3/20 0.41
PTGS2 P35354 1/20 0.41
GAA P10253 2/20 0.40
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29811842 1.00 ALDH1A1 (0.50) ALDH1A1LCKFYNKDM4ELMNA
SCHEMBL2215207 0.93 ALDH1A1 (0.50) ALDH1A1LCKFYNKDM4ELMNA
SCHEMBL7019323 0.86 KDM4E (0.51) ALDH1A1LCKFYNKDM4ELMNA
SCHEMBL3801667 0.86 KDM4E (0.47) ALDH1A1KDM4ELMNAHTTMAPK1
SCHEMBL1766160 0.85 LCK (0.60) ALDH1A1LCKFYNKDM4ELMNA
SCHEMBL2902421 0.85 ALDH1A1 (0.56) ALDH1A1LCKFYNKDM4ELMNA
SCHEMBL221470 0.84 KDM4E (0.64) ALDH1A1KDM4ELMNAHTTMAPK1
SCHEMBL9706363 0.83 ALDH1A1 (0.59) ALDH1A1LCKFYNKDM4ELMNA
SCHEMBL18669213 0.83 KDM4E (0.56) ALDH1A1LCKFYNKDM4ELMNA
SCHEMBL18700941 0.83 HTT (0.55) ALDH1A1LCKFYNKDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 158 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117164855-A High-cohesiveness branched polyimide polymer and preparation method thereof 江苏环峰电工材料有限公司 2023-12-05 CN claimed
US-20260098032-A1 METHODS AND COMPOUNDS FOR RESTORING MUTANT p53 FUNCTION PMV PHARMACEUTICALS INC (US) 2026-04-09 US disclosed
US-12594275-B2 Immunophilin binding agents and uses thereof THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2026-04-07 US disclosed
US-12558356-B2 Immunophilin binding agents and uses thereof THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2026-02-24 US disclosed
EP-4644387-A2 METHODS AND COMPOUNDS FOR RESTORING MUTANT P53 FUNCTION PMV Pharmaceuticals, Inc. (US) 2025-11-05 EP disclosed
US-12428406-B2 Methods and compounds for restoring mutant p53 function PMV PHARMACEUTICALS, INC. (US) 2025-09-30 US disclosed
US-12410187-B2 Fused tricyclic compounds useful as anticancer agents ASTRAZENECA AB (SE) 2025-09-09 US disclosed
US-20250154134-A1 COMPOUND AS FAK INHIBITOR AND USE THEREOF Wigen Biomedicine Technology (shanghai) Co., Ltd. (CN) 2025-05-15 US disclosed
US-20250108052-A1 IMMUNOPHILIN BINDING AGENTS AND USES THEREOF THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2025-04-03 US disclosed
EP-4488272-A1 COMPOUND AS FAK INHIBITOR AND USE THEREOF Wigen Biomedicine Technology (Shanghai) Co., Ltd. (CN) 2025-01-08 EP disclosed
US-20090281092-A1 POLO-LIKE KINASE INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-11-12 US disclosed
CN-101511836-A Fused pyrimido compounds ASTRAZENECA AB (SE) 2009-08-19 CN disclosed
EP-2046793-A2 FUSED PYRIMIDO COMPOUNDS AstraZeneca AB (SE) 2009-04-15 EP disclosed
WO-2009043889-A2 OXADIAZOLE DERIVATIVES MERCK SERONO S.A. (CH) 2009-04-09 WO disclosed
WO-2009042711-A1 POLO-LIKE KINASE INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-04-02 WO disclosed
WO-2009042711-A1 POLO-LIKE KINASE INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-04-02 WO disclosed
WO-2008040951-A1 COMPOUNDS ASTRAZENECA AB (SE) 2008-04-10 WO disclosed
WO-2008040951-A1 COMPOUNDS ASTRAZENECA AB (SE) 2008-04-10 WO disclosed
WO-2008003958-A2 FUSED PYRIMIDO COMPOUNDS ASTRAZENECA AB (SE) 2008-01-10 WO disclosed
US-20080009482-A1 NOVEL COMPOUNDS ASTRAZENECA AB (SE) 2008-01-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (9 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12410187-B2 Fused tricyclic compounds useful as anticancer agents MCL1, TP53, CCNA2 ALDH1A1 917/4885LCK 744/4885FYN 1350/4885
US-12594275-B2 Immunophilin binding agents and uses thereof CCR1, CCRL2, CCR3 ALDH1A1 3009/4885LCK 4015/4885FYN 3846/4885
US-12428406-B2 Methods and compounds for restoring mutant p53 function TP53, TP53BP1, KRAS ALDH1A1 1538/4885LCK 811/4885FYN 2446/4885
US-20250108052-A1 IMMUNOPHILIN BINDING AGENTS AND USES THEREOF SERPINA6, SELPLG, FABP7 ALDH1A1 3339/4885LCK 1605/4885FYN 2123/4885
US-20090281092-A1 POLO-LIKE KINASE INHIBITORS PLK1, PLK2, POLK ALDH1A1 4009/4885LCK 364/4885FYN 944/4885
US-20080009482-A1 NOVEL COMPOUNDS CYP11B2, CYP11B1, CYP46A1 ALDH1A1 422/4885LCK 4363/4885FYN 3566/4885
US-20260098032-A1 METHODS AND COMPOUNDS FOR RESTORING MUTANT p53 FUNCTION TP53, TP53BP1, MDM2 ALDH1A1 4027/4885LCK 1126/4885FYN 2355/4885
US-20250154134-A1 COMPOUND AS FAK INHIBITOR AND USE THEREOF PTK2, PAK1, FYN ALDH1A1 1905/4885LCK 21/4885FYN 3/4885
US-12558356-B2 Immunophilin binding agents and uses thereof CCRL2, CFB, CCR3 ALDH1A1 2201/4885LCK 3221/4885FYN 3393/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.