SCHEMBL2215959

SCHEMBL2215959

CCc1nc(C(=O)O)cc2c3ccccc3n(C(CC)c3ccccc3)c12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.41
GABRP O00591 1/20 0.37
GABRD O14764 1/20 0.37
GABRA1 P14867 1/20 0.37
GABRB1 P18505 1/20 0.37
GABRG2 P18507 1/20 0.37
GABRB3 P28472 1/20 0.37
GABRA5 P31644 1/20 0.37
GABRA3 P34903 1/20 0.37
GABRA2 P47869 1/20 0.37
GABRB2 P47870 1/20 0.37
GABRA4 P48169 1/20 0.37
GABRE P78334 1/20 0.37
GABRA6 Q16445 1/20 0.37
GABRG1 Q8N1C3 1/20 0.37
GABRG3 Q99928 1/20 0.37
GABRQ Q9UN88 1/20 0.37
KDM4C Q9H3R0 1/20 0.36
ALOX15 P16050 2/20 0.34
ALDH1A1 P00352 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2214017 0.91 POLB (0.40) POLBKDM4CALOX15ALDH1A1HPGD
SCHEMBL2213028 0.88 POLB (0.42) POLBKDM4CALOX15ALDH1A1HPGD
SCHEMBL2215670 0.81 CNR2 (0.43) POLBGABRPGABRDGABRA1GABRB1
SCHEMBL29217020 0.80 KDM4E (0.46) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL2214060 0.79 ALDH1A1 (0.48) POLBALOX15ALDH1A1HPGDPTGER4
SCHEMBL2215825 0.78 POLB (0.43) POLBGABRPGABRDGABRA1GABRB1
SCHEMBL2216277 0.78 CNR2 (0.43) POLBGABRPGABRDGABRA1GABRB1
SCHEMBL2214735 0.76 CYP19A1 (0.47) POLBALDH1A1HPGDKDM4EMAPK1
SCHEMBL2218129 0.75 PGR (0.47) ALDH1A1HPGD
SCHEMBL2217196 0.74 MEN1 (0.43) ALDH1A1HPGDKDM4EMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1634881-B1 HARMINE DERIVATIVES, INTERMEDIATES USED IN THEIR PREPARATION, PREPARATION PROCESSES AND USE THEREOF XINJIANG HUASHIDAN PHARMACEUTICAL RES CO LTD (CN) 2011-07-27 EP claimed