SCHEMBL22199045

SCHEMBL22199045

Cc1cn(-c2ccc(C#N)c(F)c2)cn1

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
USP30 Q70CQ3 1/20 0.47
CYP11B1 P15538 2/20 0.42
CYP11B2 P19099 2/20 0.42
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP19A1 P11511 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
CYP2E1 P05181 1/20 0.41
CYP2A6 P11509 1/20 0.41
NR2E1 Q9Y466 2/20 0.41
MAOA P21397 1/20 0.40
MAOB P27338 1/20 0.40
TRPV4 Q9HBA0 1/20 0.40
EGLN2 Q96KS0 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22199020 0.85 CYP11B2 (0.43) CYP11B1CYP11B2CYP1A2CYP3A4CYP2D6
SCHEMBL22185263 0.83 PIK3CD (0.39) CYP11B1CYP11B2TRPV4
SCHEMBL1828556 0.79 NR2E1 (0.43) CYP1A2CYP3A4CYP2D6CYP19A1CYP2C9
SCHEMBL22198918 0.76 CYP1A2 (0.46) USP30CYP1A2CYP3A4CYP2D6CYP19A1
SCHEMBL12676199 0.76 USP30 (0.40) USP30CYP1A2CYP3A4CYP2D6CYP19A1
SCHEMBL22199043 0.75 MAOA (0.53) CYP1A2CYP3A4CYP2D6CYP19A1CYP2C9
SCHEMBL1162746 0.74 CYP1A2 (0.55) USP30CYP11B2CYP1A2CYP3A4CYP2D6
SCHEMBL1903855 0.74 GRIA1 (0.42) CYP1A2
SCHEMBL2525846 0.73 CYP11B1 (0.40) CYP11B1CYP11B2TRPV4EGLN2
SCHEMBL2824888 0.73 PSEN1 (0.49) USP30

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020141439-A1 HETEROCYCLIC COMPOUNDS AS MUTANT IDH INHIBITORS INTEGRAL BIOSCIENCES PRIVATE LIMITED (IN) 2020-07-09 WO disclosed