SCHEMBL22199020

SCHEMBL22199020

Cc1cn(-c2ccc(C#N)c(C)c2)cn1

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 3/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP19A1 P11511 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
CYP2E1 P05181 1/20 0.43
CYP2A6 P11509 1/20 0.43
MAOA P21397 1/20 0.42
MAOB P27338 1/20 0.42
CYP11B1 P15538 1/20 0.41
NR2E1 Q9Y466 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22199045 0.85 USP30 (0.47) CYP11B2CYP1A2CYP3A4CYP2D6CYP19A1
SCHEMBL1828556 0.82 NR2E1 (0.43) CYP1A2CYP3A4CYP2D6CYP19A1CYP2C9
SCHEMBL24135174 0.81 CYP11B2 (0.42) CYP11B2CYP11B1
SCHEMBL9699728 0.79 NR2E1 (0.46) CYP1A2CYP3A4CYP2D6CYP19A1CYP2C9
SCHEMBL12676199 0.79 USP30 (0.40) CYP1A2CYP3A4CYP2D6CYP19A1CYP2C9
SCHEMBL1162746 0.77 CYP1A2 (0.55) CYP11B2CYP1A2CYP3A4CYP2D6CYP19A1
SCHEMBL1903855 0.76 GRIA1 (0.42) CYP1A2
SCHEMBL22198918 0.76 CYP1A2 (0.46) CYP1A2CYP3A4CYP2D6CYP19A1CYP2C9
SCHEMBL9701793 0.76 NR2E1 (0.48) CYP1A2CYP3A4CYP2D6CYP19A1CYP2C9
SCHEMBL27985278 0.75 CYP1A2 (0.65) CYP1A2CYP3A4CYP2D6CYP19A1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020141439-A1 HETEROCYCLIC COMPOUNDS AS MUTANT IDH INHIBITORS INTEGRAL BIOSCIENCES PRIVATE LIMITED (IN) 2020-07-09 WO disclosed