SCHEMBL22200410

SCHEMBL22200410

COc1cc2sc(C(F)(F)CCC(=O)NO)cc2c(F)c1OC

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
STING1 Q86WV6 6/20 0.53
HDAC1 Q13547 9/20 0.38
HDAC2 Q92769 8/20 0.38
HDAC6 Q9UBN7 6/20 0.38
HDAC3 O15379 4/20 0.38
HDAC4 P56524 4/20 0.38
HDAC7 Q8WUI4 4/20 0.38
HDAC10 Q969S8 4/20 0.38
HDAC11 Q96DB2 4/20 0.38
HDAC8 Q9BY41 4/20 0.38
HDAC9 Q9UKV0 4/20 0.38
HDAC5 Q9UQL6 4/20 0.38
TUBB4A P04350 2/20 0.36
TUBB P07437 2/20 0.36
TUBA3C P0DPH7 2/20 0.36
TUBA1B P68363 2/20 0.36
TUBA4A P68366 2/20 0.36
TUBB4B P68371 2/20 0.36
TUBB3 Q13509 2/20 0.36
TUBB2A Q13885 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22200458 0.90 STING1 (0.54) STING1TUBB1LMNASMN1; SMN2USP2
SCHEMBL22200412 0.88 STING1 (0.64) STING1SMN1; SMN2
SCHEMBL22200404 0.82 STING1 (0.48) STING1LMNAALDH1A1
SCHEMBL24175605 0.81 STING1 (0.49) STING1TUBB4ATUBBTUBA3CTUBA1B
SCHEMBL24175053 0.80 STING1 (0.49) STING1TUBB4ATUBBTUBA3CTUBA1B
SCHEMBL24175566 0.80 STING1 (0.48) STING1TUBB1USP2TSHRALDH1A1
SCHEMBL24175604 0.80 STING1 (0.54) STING1TSHRALDH1A1
SCHEMBL24175795 0.80 STING1 (0.53) STING1USP2TSHRALDH1A1
SCHEMBL22200651 0.80 STING1 (0.32) STING1
SCHEMBL22200416 0.80 STING1 (0.46) STING1HDAC1HDAC2HDAC6HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3907221-A1 FLUORINE-CONTAINING SUBSTITUTED BENZOTHIOPHENE COMPOUND, AND PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF Shanghai Institute of Materia Medica, Chinese Academy of Sciences (CN) 2021-11-10 EP disclosed
WO-2020140894-A1 FLUORINE-CONTAINING SUBSTITUTED BENZOTHIOPHENE COMPOUND, AND PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF 中国科学院上海药物研究所 2020-07-09 WO disclosed