SCHEMBL22200458

SCHEMBL22200458

COC(=O)CCC(F)(F)c1cc2c(F)c(OC)c(OC)cc2s1

nearest known ligand 0.54

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
STING1 Q86WV6 8/20 0.54
ACHE P22303 1/20 0.34
CYP3A4 P08684 2/20 0.33
CYP2C19 P33261 2/20 0.33
CYP2C9 P11712 1/20 0.33
CSNK1D P48730 1/20 0.33
ALDH1A1 P00352 3/20 0.33
LMNA P02545 2/20 0.33
HTT P42858 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
USP2 O75604 1/20 0.33
TSHR P16473 1/20 0.33
KDM4E B2RXH2 2/20 0.32
CYP1A2 P05177 1/20 0.32
TUBB1 Q9H4B7 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22200410 0.90 STING1 (0.53) STING1ALDH1A1LMNAHTTSMN1; SMN2
SCHEMBL22200412 0.89 STING1 (0.64) STING1SMN1; SMN2
SCHEMBL24175668 0.88 STING1 (0.41) STING1ACHECYP3A4CYP2C19CYP2C9
SCHEMBL22200404 0.83 STING1 (0.48) STING1ALDH1A1LMNA
SCHEMBL24175052 0.82 STING1 (0.49) STING1CYP3A4CYP2C19CYP2C9CSNK1D
SCHEMBL24175605 0.82 STING1 (0.49) STING1CYP3A4CYP2C19CYP2C9CSNK1D
SCHEMBL24175053 0.81 STING1 (0.49) STING1CYP3A4CYP2C19CYP2C9HTT
SCHEMBL24175795 0.81 STING1 (0.53) STING1CYP3A4CYP2C19CYP2C9CSNK1D
SCHEMBL24175566 0.81 STING1 (0.48) STING1CYP3A4CYP2C19CYP2C9CSNK1D
SCHEMBL24175103 0.81 STING1 (0.53) STING1CYP3A4CYP2C19CYP2C9CSNK1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022002077-A1 ARYL AROMATIC HETEROCYCLIC DERIVATIVE AND PREPARATION METHOD THEREFOR AND USE THEREOF 上海海和药物研究开发股份有限公司 2022-01-06 WO disclosed
EP-3907221-A1 FLUORINE-CONTAINING SUBSTITUTED BENZOTHIOPHENE COMPOUND, AND PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF Shanghai Institute of Materia Medica, Chinese Academy of Sciences (CN) 2021-11-10 EP disclosed
WO-2020140894-A1 FLUORINE-CONTAINING SUBSTITUTED BENZOTHIOPHENE COMPOUND, AND PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF 中国科学院上海药物研究所 2020-07-09 WO disclosed