SCHEMBL22200818

SCHEMBL22200818

Cc1nc(NSc2ccccc2C#N)ccc1-c1nc2cnc(N)nc2n(C(C)C)c1=O

nearest known ligand 0.36

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MTOR P42345 9/20 0.36
RORC P51449 1/20 0.33
PIK3CD O00329 1/20 0.32
PIK3R1 P27986 1/20 0.32
PIK3CA P42336 6/20 0.32
ERN1 O75460 1/20 0.31
ADORA2A P29274 1/20 0.30
ADORA1 P30542 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22200378 0.90 ERN1 (0.34) ERN1
SCHEMBL22200653 0.88 MTOR (0.38) MTORRORCPIK3CA
SCHEMBL22200424 0.88 MTOR (0.37) MTORRORCPIK3CA
SCHEMBL25034241 0.84 ERN1 (0.36) MTORRORCPIK3CDPIK3R1PIK3CA
SCHEMBL22200601 0.79 ERN1 (0.43) MTORPIK3CDPIK3CAERN1
SCHEMBL22200792 0.78 MTOR (0.35) MTORRORCPIK3CA
SCHEMBL22200825 0.75 CYP1A2 (0.36) MTORRORC
SCHEMBL22200739 0.75 BTK (0.43) MTORPIK3CA
SCHEMBL25034228 0.74 FEN1 (0.39) MTORRORCPIK3CA
SCHEMBL22200802 0.74 MTOR (0.41) MTORPIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020142612-A1 PYRIDO-PYRIMIDINONE AND PTERIDINONE COMPOUNDS AS INHIBITORS OF ENDORIBONUCLEASE INOSITOL REQUIRING ENZYME I (IRE I ALPHA) FOR THE TREATMENT OF CANCER DISEASES. GENENTECH, INC. (US) 2020-07-09 WO disclosed