SCHEMBL2220108

SCHEMBL2220108

Cc1nc(C(=O)O)cc2c3ccccc3n(CC(=O)c3ccccc3)c12

nearest known ligand 0.50

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.45
KMT2A Q03164 3/20 0.45
PTGER4 P35408 2/20 0.44
CTSD P07339 1/20 0.43
GPR35 Q9HC97 1/20 0.43
CYP1A2 P05177 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
KDM4E B2RXH2 1/20 0.41
MAPK1 P28482 1/20 0.41
ALDH1A1 P00352 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2214585 0.88 KMT2A (0.56) MEN1KMT2APTGER4KDM4EALDH1A1
SCHEMBL2217196 0.86 MEN1 (0.43) MEN1KMT2ACTSDGPR35CYP1A2
SCHEMBL2216231 0.85 PTGER4 (0.54) MEN1KMT2APTGER4SMN1; SMN2KDM4E
SCHEMBL2215283 0.83 CYP19A1 (0.49) MEN1KMT2ACYP1A2CYP2C9CYP2C19
SCHEMBL2215558 0.81 CNR2 (0.50) KDM4EALDH1A1
SCHEMBL2213030 0.79 SIGMAR1 (0.45) PTGER4
SCHEMBL2216044 0.79 ALDH1A1 (0.42) MEN1KMT2APTGER4SMN1; SMN2KDM4E
SCHEMBL29217034 0.79 CCR2 (0.50) MEN1KMT2ACYP1A2CYP2D6CYP2C9
SCHEMBL27899832 0.79 CNR2 (0.53)
SCHEMBL2218077 0.78 KDM4E (0.49) MEN1KMT2APTGER4KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1634881-B1 HARMINE DERIVATIVES, INTERMEDIATES USED IN THEIR PREPARATION, PREPARATION PROCESSES AND USE THEREOF XINJIANG HUASHIDAN PHARMACEUTICAL RES CO LTD (CN) 2011-07-27 EP claimed