SCHEMBL22207115

SCHEMBL22207115

CCNC(=O)c1ncc(Br)s1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.45
MAPK10 P53779 1/20 0.45
LMNA P02545 2/20 0.39
TP53 P04637 1/20 0.39
IKBKB O14920 1/20 0.39
CHUK O15111 1/20 0.39
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
PKM P14618 1/20 0.38
HDAC6 Q9UBN7 3/20 0.38
HDAC1 Q13547 2/20 0.38
HDAC4 P56524 1/20 0.38
CCNE1 P24864 1/20 0.38
CDK2 P24941 1/20 0.38
CDK5 Q00535 1/20 0.38
CNR1 P21554 1/20 0.37
HPGD P15428 1/20 0.37
FPR2 P25090 1/20 0.35
ALDH1A1 P00352 1/20 0.35
MAPT P10636 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22207107 0.80 FPR2 (0.50) SMN1; SMN2TP53NPC1RAB9AHDAC6
SCHEMBL12124304 0.80 SMYD3 (0.47) SMN1; SMN2LMNAIKBKBCHUKNPC1
SCHEMBL19951035 0.79 SMN1; SMN2 (0.41) SMN1; SMN2MAPK10LMNAIKBKBCHUK
SCHEMBL15296863 0.79 SMYD3 (0.50) SMN1; SMN2LMNATP53IKBKBCHUK
SCHEMBL17065934 0.78 ULK1 (0.44) SMN1; SMN2MAPK10LMNAHDAC6HDAC1
SCHEMBL15550220 0.75 LMNA (0.46) SMN1; SMN2MAPK10LMNANPC1RAB9A
SCHEMBL6288006 0.75 SMN1; SMN2 (0.60) SMN1; SMN2MAPK10LMNANPC1RAB9A
SCHEMBL1808824 0.74
SCHEMBL23617261 0.73 SMN1; SMN2 (0.43) SMN1; SMN2MAPK10LMNANPC1RAB9A
SCHEMBL2605695 0.72 HDAC6 (0.60) NPC1HDAC6HDAC1CCNE1CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114014854-B Dihydroisoquinoline compound 苏州爱科百发生物医药技术有限公司 2023-04-07 CN disclosed
CN-113999224-B Dihydroisoquinoline compound 苏州爱科百发生物医药技术有限公司 2023-04-07 CN disclosed
CN-114014854-A Dihydroisoquinoline compound 苏州爱科百发生物医药技术有限公司 2022-02-08 CN disclosed
CN-113999224-A Dihydroisoquinoline compound 苏州爱科百发生物医药技术有限公司 2022-02-01 CN disclosed
EP-3909951-A1 DIHYDROISOQUINOLINE COMPOUND Suzhou Ark Biopharmaceutical Co., Ltd (CN) 2021-11-17 EP disclosed
WO-2020143604-A1 DIHYDROISOQUINOLINE COMPOUND 苏州爱科百发生物医药技术有限公司 2020-07-16 WO disclosed
WO-2020143604-A1 DIHYDROISOQUINOLINE COMPOUND 苏州爱科百发生物医药技术有限公司 2020-07-16 WO disclosed
CN-111410653-A Dihydroisoquinoline compound 苏州爱科百发生物医药技术有限公司 2020-07-14 CN disclosed