SCHEMBL2221094

SCHEMBL2221094

CCCc1nc(-c2cccc(Cc3nn(-c4cc(F)cc(C#N)c4)ccc3=O)c2)n[nH]1

nearest known ligand 0.34

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 8/20 0.34
ADORA1 P30542 6/20 0.33
PGR P06401 1/20 0.32
CTSS P25774 2/20 0.32
CTSK P43235 2/20 0.32
AOC3 Q16853 2/20 0.30
NR1H2 P55055 1/20 0.30
NR1H3 Q13133 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2221088 0.81 PGR (0.33) PGR
SCHEMBL13274575 0.81 HDAC1 (0.33) ADORA2APGR
SCHEMBL2351533 0.80 MET (0.39)
SCHEMBL2268618 0.80 ADORA2A (0.35) ADORA2AADORA1NR1H2NR1H3
SCHEMBL13274793 0.79 MET (0.43)
SCHEMBL2223533 0.77 MET (0.40) CTSS
SCHEMBL13274837 0.77 MET (0.42) ADORA2A
SCHEMBL2220189 0.75 MET (0.38)
SCHEMBL12517966 0.73 MET (0.55)
SCHEMBL13274666 0.72 LMNA (0.37)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011084402-A1 TYROSINE KINASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2011-07-14 WO disclosed