Adenosine

Adenosine

SCHEMBL2221271

Nc1ncnc2c1ncn2[C@@H]1O[C@H](CO)[C@@H](O)[C@H]1O.O=C[C@H](OP(=O)(O)O)[C@@H](OP(=O)(O)O)[C@H](O)[C@H](O)CO

nearest known ligand 0.60

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ADORA1ADORA2AADORA2BADORA3

The experimentally established mechanism targets of Adenosine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 known ✓ P30542 3/20 0.60
ADORA3 known ✓ P0DMS8 2/20 0.60
ADORA2A known ✓ P29274 1/20 0.60
ADORA2B known ✓ P29275 1/20 0.60
SMN1; SMN2 Q16637 3/20 0.60
DPP4 P27487 1/20 0.60
MEN1 O00255 1/20 0.60
SLC28A1 O00337 1/20 0.60
MAP3K7 O43318 1/20 0.60
SLC28A2 O43868 1/20 0.60
GAPDH P04406 1/20 0.60
MAPK1 P28482 1/20 0.60
STAT6 P42226 1/20 0.60
PI4KA P42356 1/20 0.60
KMT2A Q03164 1/20 0.60
PI4K2B Q8TCG2 1/20 0.60
DOT1L Q8TEK3 1/20 0.60
SLC29A1 Q99808 1/20 0.60
PI4K2A Q9BTU6 1/20 0.60
SLC28A3 Q9HAS3 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Adenosine SCHEMBL472873 0.96 ADORA1 (0.63) ADORA1SMN1; SMN2ADORA3DPP4MEN1
Adenosine SCHEMBL16762258 0.89 P2RY2 (0.63) ADORA1SMN1; SMN2ADORA3DPP4MEN1
Adenosine SCHEMBL3485281 0.87 ADORA1 (0.48) ADORA1SMN1; SMN2ADORA3DPP4MEN1
Adenosine SCHEMBL9419203 0.87 ADORA1 (0.63) ADORA1SMN1; SMN2ADORA3DPP4MEN1
Adenosine SCHEMBL28057366 0.86 ADORA1 (0.67) ADORA1SMN1; SMN2ADORA3DPP4MEN1
Adenosine SCHEMBL27686613 0.86 P2RY2 (0.65) ADORA1SMN1; SMN2ADORA3DPP4MEN1
Guanosine SCHEMBL6027663 0.85 NT5E (0.55) NT5E
Guanosine SCHEMBL7571212 0.85 NT5E (0.55) NT5E
Adenosine SCHEMBL2327105 0.84 ADORA3 (0.72) ADORA1SMN1; SMN2ADORA3DPP4MEN1
Adenosine SCHEMBL26612876 0.84 ADORA3 (0.72) ADORA1SMN1; SMN2ADORA3DPP4MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 36 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250075170-A1 TARGETED MUTAGENESIS IN SPIRULINA Lumen Bioscience, Inc. 2025-03-06 US disclosed
US-12065638-B2 Targeted mutagenesis in spirulina Lumen Bioscience, Inc. (US) 2024-08-20 US disclosed
EP-3191581-B9 TARGETED MUTAGENESIS IN SPIRULINA LUMEN BIOSCIENCE INC (US) 2023-10-11 EP disclosed
EP-3191581-B1 TARGETED MUTAGENESIS IN SPIRULINA LUMEN BIOSCIENCE INC (US) 2023-06-07 EP disclosed
US-20230080657-A1 METHODS FOR NUCLEIC ACID SEQUENCING SARMAL, INC. 2023-03-16 US disclosed
EP-4085153-A2 METHODS FOR NUCLEIC ACID SEQUENCING Sarmal, Inc. (US) 2022-11-09 EP disclosed
US-20180148732-A1 METHODS OF MODIFYING OIL CONTENT IN PLANTS AND PLANTS PRODUCED THEREBY THE STATE OF ISRAEL, MINISTRY OF AGRICULTURE & RURAL DEVELOPMENT, AGRICULTURAL RESEARCH ORGANIZATION (ARO) (VOLCANI CENTER) (IL) 2018-05-31 US disclosed
US-9914947-B2 Biological production of organic compounds ALLIANCE FOR SUSTAINABLE ENERGY, LLC (US) 2018-03-13 US disclosed
US-20160177353-A1 BIOLOGICAL PRODUCTION OF ORGANIC COMPOUNDS Alliance for Energy Innovation, LLC 2016-06-23 US disclosed
US-9309541-B2 Biological production of organic compounds ALLIANCE FOR SUSTAINABLE ENERGY, LLC (US) 2016-04-12 US disclosed
WO-2002103001-A1 GDP-MANNOSE-3',5'-EPIMERASE AND METHODS OF USE THEREOF VLAAMS INTERUNIVERSITAIR INSTITUUT VOOR BIOTECHNOLOGIE VZW (BE) 2002-12-27 WO disclosed
US-6486383-B1 Modification of starch content in plants ADVANCED TECHNOLOGIES (CAMBRIDGE) LIMITED (GB) 2002-11-26 US disclosed
EP-1150709-A2 ANTI-MICROBIAL AGENTS, DIAGNOSTIC REAGENTS, AND VACCINES BASED ON APICOMPLEXAN PARASITE COMPONENTS Mcleod, Rima W. (US) 2001-11-07 EP disclosed
WO-2000066154-A2 ANTI-MICROBIAL AGENTS, DIAGNOSTIC REAGENTS, AND VACCINES BASED ON UNIQUE APICOMPLEXAN PARASITE COMPONENTS ARCH DEVELOPMENT CORPORATION (US) 2000-11-09 WO disclosed
US-6096945-A AMPLIFICATION OF PHOSPHORYLASE ACTIVITY IN MAIZE, WHEAT, RICE, POTATO, PEAS, PEANUT, CASSAVA, BEANS, CARROTS, TOMATO AND TOBACCO; INSERTION OF GENE CODING A PEPTIDE CHAIN OF PHOSPHORYLASE, SCREEN FOR AMPLIFIED GENE EXPRESSION IN PLANTS ADVANCED TECHNOLOGIES (CAMBRIDGE) LIMITED (GB) 2000-08-01 US disclosed
WO-1998003661-A9 ANTIMICROBIAL AGENTS, DIAGNOSTIC REAGENTS, AND VACCINES BASED ON UNIQUE APICOMPLEXAN PARASITE COMPONENTS 1998-05-28 WO disclosed
EP-0772682-A1 MODIFICATION OF STARCH CONTENT IN PLANTS ADVANCED TECHNOLOGIES (CAMBRIDGE) LIMITED (GB) 1997-05-14 EP disclosed
EP-0772682-A1 MODIFICATION OF STARCH CONTENT IN PLANTS ADVANCED TECHNOLOGIES (CAMBRIDGE) LIMITED (GB) 1997-05-14 EP disclosed
WO-1995034660-A1 MODIFICATION OF STARCH CONTENT IN PLANTS ADVANCED TECHNOLOGIES (CAMBRIDGE) LIMITED (GB) 1995-12-21 WO disclosed
WO-1995034660-A1 MODIFICATION OF STARCH CONTENT IN PLANTS ADVANCED TECHNOLOGIES (CAMBRIDGE) LIMITED (GB) 1995-12-21 WO disclosed