Adenosine

Adenosine

SCHEMBL472873

Nc1ncnc2c1ncn2[C@@H]1O[C@H](CO)[C@@H](O)[C@H]1O.O=C[C@H](OP(=O)(O)O)[C@H](OP(=O)(O)O)[C@H](O)CO

nearest known ligand 0.63

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ADORA1ADORA2AADORA2BADORA3

The experimentally established mechanism targets of Adenosine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 known ✓ P30542 3/20 0.63
ADORA3 known ✓ P0DMS8 2/20 0.63
ADORA2A known ✓ P29274 1/20 0.63
ADORA2B known ✓ P29275 1/20 0.63
SMN1; SMN2 Q16637 3/20 0.63
DPP4 P27487 1/20 0.63
MEN1 O00255 1/20 0.63
SLC28A1 O00337 1/20 0.63
MAP3K7 O43318 1/20 0.63
SLC28A2 O43868 1/20 0.63
GAPDH P04406 1/20 0.63
MAPK1 P28482 1/20 0.63
STAT6 P42226 1/20 0.63
PI4KA P42356 1/20 0.63
KMT2A Q03164 1/20 0.63
PI4K2B Q8TCG2 1/20 0.63
DOT1L Q8TEK3 1/20 0.63
SLC29A1 Q99808 1/20 0.63
PI4K2A Q9BTU6 1/20 0.63
SLC28A3 Q9HAS3 1/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Adenosine SCHEMBL2221271 0.96 ADORA1 (0.60) ADORA1SMN1; SMN2ADORA3DPP4MEN1
Adenosine SCHEMBL16762258 0.88 P2RY2 (0.63) ADORA1SMN1; SMN2ADORA3DPP4MEN1
Adenosine SCHEMBL9419203 0.85 ADORA1 (0.63) ADORA1SMN1; SMN2ADORA3DPP4MEN1
Adenosine SCHEMBL10980572 0.85 ADORA1 (0.74) ADORA1SMN1; SMN2ADORA3DPP4MEN1
Adenosine SCHEMBL28057366 0.85 ADORA1 (0.67) ADORA1SMN1; SMN2ADORA3DPP4MEN1
Adenosine SCHEMBL27686613 0.85 P2RY2 (0.65) ADORA1SMN1; SMN2ADORA3DPP4MEN1
Adenosine SCHEMBL26612876 0.83 ADORA3 (0.72) ADORA1SMN1; SMN2ADORA3DPP4MEN1
Adenosine SCHEMBL2327105 0.83 ADORA3 (0.72) ADORA1SMN1; SMN2ADORA3DPP4MEN1
Adenosine SCHEMBL28186074 0.83 P2RY2 (0.80) ADORA1SMN1; SMN2ADORA3DPP4MEN1
Adenosine SCHEMBL30301161 0.82 ADORA1 (0.81) ADORA1SMN1; SMN2ADORA3DPP4MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 66 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220241416-A1 METHODS FOR THE IDENTIFICATION OF SARM1 NADASE ACTIVITY INHIBITORS AND USES THEREOF UNIV BAR ILAN (US) 2022-08-04 US claimed
EP-4592305-A2 PRODUCTION OF CYCLIC ADENYLATES AND THEIR USE AS ALLOSTERIC REGULATORS Vilnius University (LT) 2025-07-30 EP disclosed
US-12370209-B2 Methods for the use of 5′-adenosine diphosphate ribose (ADPR) INVIRSA, INC. (US) 2025-07-29 US disclosed
WO-2025122455-A1 METHODS FOR THE USE OF 5'-ADENOSINE DIPHOSPHATE RIBOSE (ADPR) FOR VEGF MODULATION INVIRSA, INC. (US) 2025-06-12 WO disclosed
US-20250161343-A1 METHODS FOR THE USE OF 5'-ADENOSINE DIPHOSPHATE RIBOSE (ADPR) INVIRSA, INC. (US) 2025-05-22 US disclosed
EP-3630966-B1 PRODUCTION OF CYCLIC ADENYLATES AND THEIR USE AS ALLOSTERIC REGULATORS UNIV VILNIUS (LT) 2025-04-23 EP disclosed
US-12233083-B2 Methods for the use of 5′-adenosine diphosphate ribose (ADPR) INVIRSA, INC. (US) 2025-02-25 US disclosed
US-20250020654-A1 SCREENING METHODS FOR PARP MODULATORS RIBON THERAPEUTICS, INC. 2025-01-16 US disclosed
US-12123031-B2 Regulation of CRISPR-associated rossman fold (CARF) domain containing proteins by oligoadenylates VILNIUS UNIVERSITY (LT) 2024-10-22 US disclosed
US-20240229012-A9 SITE-SPECIFIC GENOME MODIFICATION TECHNOLOGY NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2024-07-11 US disclosed
US-20030153559-A1 Propenecarboxylic acid amidoxime derivatives, a process for the preparation thereof , and pharmaceutical compositions containing the same N-GENE RESEARCH LABORATORIES INC. 2003-08-14 US disclosed
EP-1154998-A1 INHIBITORS OF CELLULAR NIACINAMIDE MONONUCLEOTIDE FORMATION AND THEIR USE IN CANCER THERAPY Klinge Pharma GmbH (DE) 2001-11-21 EP disclosed
WO-2000050399-A1 INHIBITORS OF CELLULAR NIACINAMIDE MONONUCLEOTIDE FORMATION AND THEIR USE IN CANCER THERAPY KLINGE PHARMA GMBH (DE) 2000-08-31 WO disclosed
EP-0918789-A1 PYRIDINE NUCLEOTIDE-DEPENDENT ENZYMES THE UNIVERSITY OF SHEFFIELD (GB) 1999-06-02 EP disclosed
WO-1997048722-A1 PYRIDINE NUCLEOTIDE-DEPENDENT ENZYMES THE UNIVERSITY OF SHEFFIELD (GB) 1997-12-24 WO disclosed
WO-1992010198-A1 IMMUNOTHERAPEUTIC AGENTS, COMPOSITIONS AND METHODS JOHNSON & JOHNSON RESEARCH PTY LIMITED (AU) 1992-06-25 WO disclosed
EP-0090405-B1 NOVEL AZOLE DINUCLEOTIDE COMPOUNDS AND METHODS FOR THEIR PRODUCTION BRIGHAM YOUNG UNIVERSITY (US) 1986-06-25 EP disclosed
US-4594415-A Viricides ROBINS ROLAND K (US) 1986-06-10 US disclosed
US-4544741-A Azole dinucleotide compounds and methods for their production BRIGHAM YOUNG UNIVERSITY, PROVO, UT., A NONPROFIT CORP. OF UT 1985-10-01 US disclosed
EP-0090405-A1 Novel azole dinucleotide compounds and methods for their production BRIGHAM YOUNG UNIVERSITY (US) 1983-10-05 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12370209-B2 Methods for the use of 5′-adenosine diphosphate ribose (ADPR) ADAR, CD38, PARP1 ADORA1 22/4885ADORA3 21/4885ADORA2A 6/4885
US-20250161343-A1 METHODS FOR THE USE OF 5'-ADENOSINE DIPHOSPHATE RIBOSE (ADPR) SIRT6, ADAR, SIRT1 ADORA1 157/4885ADORA3 112/4885ADORA2A 59/4885
US-12233083-B2 Methods for the use of 5′-adenosine diphosphate ribose (ADPR) SIRT6, ADAR, SIRT1 ADORA1 168/4885ADORA3 125/4885ADORA2A 63/4885
US-20030153559-A1 Propenecarboxylic acid amidoxime derivatives, a process for the preparation thereof , and pharmaceutical compositions containing the same PARP1, PARP2, PARP3 ADORA1 268/4885ADORA3 196/4885ADORA2A 94/4885
US-20250020654-A1 SCREENING METHODS FOR PARP MODULATORS PARP1, PARP2, PARP3 ADORA1 2658/4885ADORA3 1428/4885ADORA2A 951/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.