SCHEMBL2221753

SCHEMBL2221753

CN(C)C(=O)C(CCN1CCC(O)CC1)(c1ccccc1)c1ccccc1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 19/20 0.71
DRD3 P35462 13/20 0.59
DRD2 P14416 12/20 0.59
DRD4 P21917 7/20 0.59
OPRD1 P41143 3/20 0.59
MEN1 O00255 2/20 0.59
LMNA P02545 2/20 0.59
ADRB2 P07550 2/20 0.59
ADRA2A P08913 2/20 0.59
SLC6A4 P31645 2/20 0.59
OPRK1 P41145 2/20 0.59
HTR2B P41595 2/20 0.59
SLC6A3 Q01959 2/20 0.59
KMT2A Q03164 2/20 0.59
SMN1; SMN2 Q16637 2/20 0.59
SIGMAR1 Q99720 2/20 0.59
SCN1A P35498 2/20 0.59
SCN2A Q99250 2/20 0.59
SCN3A Q9NY46 2/20 0.59
CES2 O00748 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1492481 0.85 OPRM1 (0.63) OPRM1DRD3DRD2DRD4OPRD1
SCHEMBL6842012 0.83 OPRM1 (0.60) OPRM1DRD3DRD2DRD4OPRD1
SCHEMBL9790173 0.83 OPRM1 (0.58) OPRM1DRD3DRD2DRD4OPRD1
SCHEMBL2571840 0.83 OPRM1 (1.00) OPRM1DRD3DRD2DRD4OPRD1
SCHEMBL6836914 0.82 OPRM1 (0.69) OPRM1DRD3DRD2DRD4OPRD1
Bromide SCHEMBL8206195 0.82 OPRM1 (0.58) OPRM1DRD3DRD2DRD4OPRD1
SCHEMBL6841059 0.81 OPRM1 (0.57) OPRM1DRD3DRD2DRD4OPRD1
SCHEMBL6841483 0.79 OPRM1 (0.55) OPRM1DRD3DRD2DRD4OPRD1
SCHEMBL9721660 0.79 OPRM1 (0.52) OPRM1DRD3DRD2DRD4OPRD1
SCHEMBL9721502 0.79 OPRM1 (0.52) OPRM1DRD3DRD2DRD4OPRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2521711-A1 QUATERNARY AMMONIUM SALT PRODRUGS Alkermes, Inc. (US) 2012-11-14 EP disclosed
WO-2011084846-A1 QUATERNARY AMMONIUM SALT PRODRUGS ALKERMES, INC. (US) 2011-07-14 WO disclosed