SCHEMBL2222752

SCHEMBL2222752

C[S+]([O-])c1ccc(N2CCC(CCN3CCCCC3)CC2)c(NC(=O)c2cccc(Cl)c2)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.52
MEN1 O00255 1/20 0.52
WDR5 P61964 1/20 0.49
GAA P10253 2/20 0.47
CXCR3 P49682 6/20 0.47
TDP1 Q9NUW8 2/20 0.45
LMNA P02545 2/20 0.45
MAPT P10636 1/20 0.45
KCNH2 Q12809 1/20 0.45
CACNA1I Q9P0X4 1/20 0.45
HTT P42858 2/20 0.44
MCL1 Q07820 1/20 0.44
APOBEC3A P31941 1/20 0.43
APOBEC3G Q9HC16 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
NPC1 O15118 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12515553 0.92 MEN1 (0.52) KMT2AMEN1WDR5GAACXCR3
SCHEMBL2221639 0.89 KMT2A (0.60) KMT2AMEN1WDR5GAACXCR3
SCHEMBL2222665 0.87 MEN1 (0.56) KMT2AMEN1WDR5GAACXCR3
SCHEMBL2222754 0.86 KMT2A (0.52) KMT2AMEN1WDR5GAACXCR3
SCHEMBL2221503 0.85 MEN1 (0.56) KMT2AMEN1WDR5GAACXCR3
SCHEMBL2221486 0.85 MEN1 (0.72) KMT2AMEN1GAACXCR3MAPT
SCHEMBL2221797 0.85 KMT2A (0.53) KMT2AMEN1WDR5GAACXCR3
SCHEMBL2220801 0.85 WDR5 (0.54) KMT2AMEN1WDR5GAACXCR3
SCHEMBL2222538 0.85 MEN1 (0.55) KMT2AMEN1WDR5GAACXCR3
SCHEMBL2221554 0.85 MEN1 (0.55) KMT2AMEN1WDR5GAACXCR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011084985-A1 CXCR3 RECEPTOR ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2011-07-14 WO claimed